SCHEMBL8990623

SCHEMBL8990623

CCOc1nc(Cc2ccc(Cl)cc2)nc(O)c1NC(=O)c1ccco1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.47
HPGD P15428 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
RAB9A P51151 4/20 0.46
NPC1 O15118 3/20 0.46
TP53 P04637 2/20 0.46
ALDH1A1 P00352 4/20 0.46
TSHR P16473 3/20 0.46
HTT P42858 1/20 0.46
MAPT P10636 4/20 0.44
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
HSD17B10 Q99714 2/20 0.43
NPSR1 Q6W5P4 1/20 0.43
NOD2 Q9HC29 1/20 0.43
NOD1 Q9Y239 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
LMNA P02545 3/20 0.42
POLB P06746 1/20 0.42
KCNMA1 Q12791 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8990578 0.81 RAB9A (0.53) KDM4EHPGDSMN1; SMN2RAB9ANPC1
SCHEMBL14552907 0.66 EGLN1 (0.44) KDM4EHPGDSMN1; SMN2RAB9ATP53
SCHEMBL655417 0.66 RAB9A (0.51) KDM4ESMN1; SMN2RAB9ANPC1TP53
SCHEMBL8990610 0.65 NPC1 (0.52) KDM4ESMN1; SMN2RAB9ANPC1TP53
SCHEMBL6632968 0.65 RAB9A (1.00) KDM4EHPGDSMN1; SMN2RAB9ANPC1
Hydrochloric Acid SCHEMBL1832732 0.65 NPC1 (0.53) KDM4ESMN1; SMN2RAB9ANPC1TP53
SCHEMBL27954065 0.65 MAPK1 (0.44) TP53MAPTPOLB
SCHEMBL8990595 0.64 RAB9A (0.50) KDM4EHPGDSMN1; SMN2RAB9ANPC1
SCHEMBL5692749 0.64 NPC1 (0.52) KDM4EHPGDSMN1; SMN2RAB9ANPC1
SCHEMBL5692659 0.63 HSD17B10 (0.68) KDM4EHPGDSMN1; SMN2RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5500428-A Furyl-substituted purines and adenosine antagonists IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1996-03-19 US disclosed
US-5300509-A Adenosine antagonists for treating cardiovascular disorders, vasodilation IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-04-05 US disclosed
EP-0544445-A2 Furyl-substituted purines, oxazolopyrimidines and pteridines as adenosine antagonists ZENECA LIMITED (GB) 1993-06-02 EP disclosed