SCHEMBL8991033

SCHEMBL8991033

CCCCCc1ccc(CCc2ccc(-c3ccc(C#N)cc3)cc2)c(F)c1

nearest known ligand 0.68

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.68
HSD17B10 Q99714 1/20 0.68
RARB P10826 8/20 0.45
RARA P10276 2/20 0.45
RARG P13631 1/20 0.45
HRH3 Q9Y5N1 4/20 0.43
S1PR1 P21453 1/20 0.40
CYP19A1 P11511 3/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
MTOR P42345 1/20 0.39
KMT2A Q03164 1/20 0.39
HTR2A P28223 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8990697 0.91 TSHR (0.52) TSHRHSD17B10HRH3CYP19A1MEN1
SCHEMBL9663375 0.86 RARB (0.51) TSHRHSD17B10RARBRARARARG
SCHEMBL8990742 0.85 RARB (0.50) TSHRHSD17B10RARBRARARARG
SCHEMBL8380924 0.85 HSD17B10 (0.93) TSHRHSD17B10RARBRARAHRH3
SCHEMBL8376946 0.85 HSD17B10 (0.93) TSHRHSD17B10RARBRARAHRH3
SCHEMBL9399089 0.85 HTR2A (0.52) HSD17B10RARBRARARARGS1PR1
SCHEMBL9398851 0.85 HTR2A (0.52) HSD17B10RARBRARARARGS1PR1
SCHEMBL9715240 0.83 HSD17B10 (0.97) TSHRHSD17B10RARBRARAHRH3
SCHEMBL9715655 0.83 HSD17B10 (0.97) TSHRHSD17B10RARBRARAHRH3
SCHEMBL508855 0.83 HSD17B10 (0.96) TSHRHSD17B10RARBRARAHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5496499-A Biphenylethanes and liquid-crystalline phase MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-03-05 US disclosed
EP-0429558-B1 DIPHENYLYLETHANES AND LIQUID CRYSTALLINE PHASE MERCK PATENT GMBH (DE) 1994-03-30 EP disclosed