SCHEMBL8990697

SCHEMBL8990697

CCCc1ccc(CCc2ccc(-c3ccc(C#N)cc3)cc2)c(F)c1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.52
HSD17B10 Q99714 1/20 0.52
HRH3 Q9Y5N1 7/20 0.45
CYP2A6 P11509 1/20 0.41
KIF11 P52732 1/20 0.39
NSD2 O96028 1/20 0.37
MMP12 P39900 1/20 0.37
MMP13 P45452 1/20 0.37
KDM1A O60341 1/20 0.37
MAPT P10636 2/20 0.37
POLB P06746 1/20 0.37
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
KMT2A Q03164 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
CYP19A1 P11511 1/20 0.36
KDM4E B2RXH2 1/20 0.36
FFAR1 O14842 1/20 0.36
FFAR4 Q5NUL3 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8991033 0.91 TSHR (0.68) TSHRHSD17B10HRH3MAPTMEN1
SCHEMBL9664336 0.88 ALOX5 (0.41) HSD17B10MAPT
SCHEMBL8990636 0.84 MAOB (0.47) HSD17B10MAPTALDH1A1
SCHEMBL9664848 0.84 TAAR1 (0.40) HSD17B10MAPT
SCHEMBL9317548 0.83 TSHR (0.71) TSHRHSD17B10HRH3CYP2A6KIF11
SCHEMBL8379783 0.83 TSHR (0.71) TSHRHSD17B10HRH3CYP2A6KIF11
SCHEMBL17108410 0.83 TSHR (0.51) TSHRHSD17B10HRH3CYP2A6KIF11
SCHEMBL9664166 0.82 RARB (0.46) TSHRHSD17B10MAPTMEN1ALDH1A1
SCHEMBL9664954 0.82 RARB (0.47) HSD17B10KIF11MAPT
SCHEMBL2041798 0.82 TSHR (0.73) TSHRHSD17B10HRH3CYP2A6KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5496499-A Biphenylethanes and liquid-crystalline phase MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-03-05 US disclosed
EP-0429558-B1 DIPHENYLYLETHANES AND LIQUID CRYSTALLINE PHASE MERCK PATENT GMBH (DE) 1994-03-30 EP disclosed