SCHEMBL8992520

SCHEMBL8992520

CCCc1nc(CO)c[nH]1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.33
ADORA2A P29274 2/20 0.33
ADORA1 P30542 2/20 0.33
GLA P06280 1/20 0.31
CCR1 P32246 1/20 0.30
BACE1 P56817 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL152356 0.89 HRH3 (0.39)
Hydrochloric Acid SCHEMBL9594946 0.87 HRH3 (0.38)
SCHEMBL2054377 0.87 GPR84 (0.41)
SCHEMBL11470771 0.85 GPR84 (0.43)
SCHEMBL3286058 0.85 BACE1 (0.36) GLABACE1
SCHEMBL674184 0.83
SCHEMBL3697323 0.83 GLA (0.33) GLABACE1
SCHEMBL3099997 0.81
SCHEMBL9937448 0.80 SMN1; SMN2 (0.32) GLABACE1
SCHEMBL3841860 0.80 HRH3 (0.41) GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0531876-B1 Imidazoindolizine derivatives and process for preparation thereof TANABE SEIYAKU CO (JP) 1996-12-18 EP disclosed
US-5510354-A HYPOTENSIVE AGENTS TANABE SEIYAKU CO., LTD. (JP) 1996-04-23 US disclosed
US-5424316-A Imidazopyridine derivatives for the treatment of hypertension TANABE SEIYAKU CO., LTD. (JP) 1995-06-13 US disclosed
US-5409936-A Useful in prophylaxix; exhibits potent angiotensin ii inhibitory acivities TANABE SEIYAKU CO., LTD. (JP) 1995-04-25 US disclosed
US-5268377-A Imidazoindolizine derivatives process for preparation thereof and use thereof to treat hypertension TANABE SEIYAKU CO., LTD. (JP) 1993-12-07 US disclosed
US-5266704-A Process for production of 2-substituted-4-hydromethylimidazole compounds NIPPON GOHSEI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1993-11-30 US disclosed
EP-0531876-A2 Imidazoindolizine derivatives and process for preparation thereof TANABE SEIYAKU CO., LTD. (JP) 1993-03-17 EP disclosed
EP-0531874-A1 Imidazopyridine derivatives and process for preparation thereof TANABE SEIYAKU CO., LTD. (JP) 1993-03-17 EP disclosed
US-RE30511-E ENZYME INHIBITOR, HERBICIDE, CYCLIZATION AMERICAN CYANAMID COMPANY (US) 1981-02-10 US disclosed
US-4168964-A HERBICIDES AMERICAN CYANAMID COMPANY (US) 1979-09-25 US disclosed
US-4124766-A INTERMEDIATES FOR PHOSPHODIESTERASE INHIBITORS AMERICAN CYANAMID COMPANY (US) 1978-11-07 US disclosed
US-4107308-A HYPOTENSIVE AGENTS, HERBICIDES, REACTING SODIUM SALT WITH ALLYL OR ALKYL HALIDE, RING CLOSURE AMERICAN CYANAMID COMPANY (US) 1978-08-15 US disclosed
US-4107307-A ENZYME INHIBITORS, HERBICIDES, RING CLOSURE AMERICAN CYANAMID COMPANY (US) 1978-08-15 US disclosed