SCHEMBL8992885

SCHEMBL8992885

N#CCc1ccc(Cc2ccc3c(c2)OCO3)cc1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.51
TAAR1 Q96RJ0 4/20 0.49
MIF P14174 1/20 0.47
SLC6A4 P31645 3/20 0.47
CYP3A4 P08684 2/20 0.47
CYP1A2 P05177 1/20 0.47
MAPT P10636 1/20 0.47
CYP2D6 P10635 2/20 0.46
SLC6A2 P23975 2/20 0.46
SLC6A3 Q01959 2/20 0.46
PIK3CA P42336 1/20 0.46
PIK3CG P48736 1/20 0.46
CMA1 P23946 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL141712 0.90 TAAR1 (0.55) HTTTAAR1MIFSLC6A4CYP3A4
SCHEMBL29358232 0.90 TAAR1 (0.55) HTTTAAR1MIFSLC6A4CYP3A4
SCHEMBL108109 0.86 TAAR1 (0.62) TAAR1MIFSLC6A4CYP3A4CYP1A2
SCHEMBL109195 0.84 TAAR1 (0.64) TAAR1MIFSLC6A4CYP3A4CYP1A2
SCHEMBL31739246 0.83 GSK3A (0.51) HTTTAAR1MIFSLC6A4CYP3A4
SCHEMBL2963428 0.83 TAAR1 (0.49) HTTTAAR1MIFSLC6A4CYP3A4
SCHEMBL1422874 0.79 ALDH1A1 (0.58) TAAR1SLC6A4CYP3A4CYP1A2MAPT
SCHEMBL1464785 0.79 CD274 (0.50) HTTTAAR1MIFSLC6A4CYP3A4
SCHEMBL11092660 0.77 CYP3A4 (0.62) TAAR1SLC6A4CYP3A4CYP1A2MAPT
SCHEMBL8993266 0.77 TAAR1 (0.53) TAAR1SLC6A4CYP3A4CYP1A2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed