SCHEMBL8992993

SCHEMBL8992993

CCOC(=O)c1cnc2c(-c3ccc(Cc4ccccc4)cc3)cnn2c1O

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.68
RAB9A P51151 5/20 0.68
SMN1; SMN2 Q16637 3/20 0.68
NFKB1 P19838 2/20 0.68
NFKB2 Q00653 2/20 0.68
RELA Q04206 2/20 0.68
MAPT P10636 2/20 0.68
ALDH1A1 P00352 3/20 0.66
KDM4E B2RXH2 3/20 0.66
TP53 P04637 1/20 0.66
HPGD P15428 1/20 0.66
STAT1 P42224 1/20 0.66
HSD17B10 Q99714 1/20 0.66
LMNA P02545 1/20 0.60
POLB P06746 1/20 0.60
GAA P10253 1/20 0.56
GPR119 Q8TDV5 11/20 0.51
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
TSHR P16473 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8992991 0.91 NPC1 (0.57) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL8993226 0.89 NPC1 (0.54) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL9168201 0.87 NPC1 (0.67) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL8992938 0.86 NPC1 (0.66) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL8992832 0.86 RAB9A (0.52) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL8993204 0.84 SMN1; SMN2 (0.52) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL4709877 0.81 NPC1 (0.59) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL11779261 0.81 NPC1 (0.66) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL8993229 0.80 BRS3 (0.52) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL8993100 0.80 NPC1 (0.53) NPC1RAB9ASMN1; SMN2NFKB1NFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed