SCHEMBL8993022

SCHEMBL8993022

CCCC(c1ccccc1)c1ccc(CC#N)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 7/20 0.41
HRH1 P35367 7/20 0.39
SIGMAR1 Q99720 1/20 0.39
KMT2A Q03164 1/20 0.37
UBE2M P61081 1/20 0.37
DCUN1D1 Q96GG9 1/20 0.37
CYP19A1 P11511 1/20 0.37
AOC3 Q16853 1/20 0.37
PBRM1 Q86U86 1/20 0.36
CCR2 P41597 1/20 0.36
HTR1A P08908 2/20 0.36
ADORA3 P0DMS8 2/20 0.36
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36
ADRA1A P35348 2/20 0.36
OPRM1 P35372 2/20 0.36
DRD3 P35462 2/20 0.36
SLC6A3 Q01959 2/20 0.36
KCNH2 Q12809 2/20 0.36
CHRM2 P08172 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8992978 0.80 MAOB (0.42) SIGMAR1KMT2APBRM1MAOB
SCHEMBL107889 0.79 HRH1 (0.56) HTR2AHRH1SIGMAR1KMT2AAOC3
SCHEMBL19113570 0.77 ESR1 (0.46) KMT2AUBE2MDCUN1D1DRD3ADRA2A
Hydrochloric Acid SCHEMBL6521685 0.77 HRH1 (0.54) HTR2AHRH1SIGMAR1KMT2AAOC3
Hydrogen Peroxide SCHEMBL27864054 0.77 HRH1 (0.54) HTR2AHRH1SIGMAR1KMT2AAOC3
Ammonia Solution, Strong SCHEMBL5724927 0.77 HRH1 (0.54) HTR2AHRH1SIGMAR1KMT2AAOC3
SCHEMBL28229621 0.77 HRH1 (0.54) HTR2AHRH1SIGMAR1KMT2AAOC3
SCHEMBL8992781 0.77 HTR2A (0.44) HTR2AHRH1SIGMAR1KMT2ACYP19A1
SCHEMBL10585427 0.77 TSHR (0.45) KMT2APBRM1LMNA
SCHEMBL10567235 0.77 TRPA1 (0.45) HTR2AKMT2APBRM1LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed