SCHEMBL8993068

SCHEMBL8993068

N#CCc1ccc(C(C=O)c2ccccc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.41
L3MBTL1 Q9Y468 1/20 0.36
MEN1 O00255 1/20 0.36
NPC1 O15118 2/20 0.33
PKM P14618 1/20 0.33
TRPA1 O75762 1/20 0.33
PBRM1 Q86U86 1/20 0.33
TSHR P16473 1/20 0.33
THRB P10828 1/20 0.33
RAB9A P51151 1/20 0.33
MAPT P10636 2/20 0.33
FLT3 P36888 1/20 0.33
ABCB1 P08183 1/20 0.33
ABCG2 Q9UNQ0 1/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
MAOB P27338 1/20 0.33
KDM4E B2RXH2 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
FFAR1 O14842 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL193931 0.77 CYP2D6 (0.48) KMT2ATSHRMAPTLMNAKDM4E
SCHEMBL10585427 0.77 TSHR (0.45) KMT2AL3MBTL1MEN1NPC1TRPA1
SCHEMBL10567235 0.77 TRPA1 (0.45) KMT2AMEN1NPC1PKMTRPA1
SCHEMBL8992978 0.77 MAOB (0.42) KMT2AL3MBTL1MEN1NPC1TRPA1
SCHEMBL5084681 0.77 TSHR (0.48) KMT2AL3MBTL1PKMTSHRMAPT
SCHEMBL11449880 0.75 ESR1 (0.37) KMT2AL3MBTL1MEN1NPC1PKM
Acetaldehyde SCHEMBL1720078 0.74 KMT2A (0.43) KMT2AL3MBTL1MEN1NPC1THRB
SCHEMBL8993022 0.72 HTR2A (0.41) KMT2APBRM1LMNAMAOBCYP2D6
SCHEMBL10564457 0.72 MAOB (0.42) KMT2AMEN1NPC1TRPA1PBRM1
SCHEMBL7042455 0.72 EPHX1 (0.49) KMT2AL3MBTL1MEN1HTTMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed