SCHEMBL8993223

SCHEMBL8993223

COC(=O)c1ccc(C(O)c2cccc(OC)c2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.55
RAB9A P51151 4/20 0.55
SMN1; SMN2 Q16637 4/20 0.55
TP53 P04637 3/20 0.55
MAPK1 P28482 2/20 0.55
ALDH1A1 P00352 2/20 0.55
PKM P14618 2/20 0.55
KMT2A Q03164 2/20 0.55
MEN1 O00255 1/20 0.55
HPGD P15428 1/20 0.55
CA1 P00915 2/20 0.53
CA2 P00918 2/20 0.53
POLB P06746 1/20 0.52
BLM P54132 1/20 0.52
AOC3 Q16853 1/20 0.51
LMNA P02545 1/20 0.51
MAPT P10636 1/20 0.51
HTT P42858 1/20 0.51
CA12 O43570 1/20 0.50
CA9 Q16790 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8993107 0.85 NPC1 (0.55) NPC1RAB9ASMN1; SMN2TP53MAPK1
SCHEMBL1894316 0.85 CA1 (0.57) CA1CA2LMNAMAPTCA12
SCHEMBL28823597 0.84 CA1 (0.75) NPC1KMT2AMEN1CA1CA2
SCHEMBL6343583 0.84 SMN1; SMN2 (0.57) NPC1RAB9ASMN1; SMN2TP53MAPK1
SCHEMBL9149153 0.84 TDP1 (0.51) RAB9AALDH1A1KMT2AMEN1CA1
SCHEMBL12019562 0.83 OPRM1 (0.50) SMN1; SMN2ALDH1A1HPGDAOC3L3MBTL1
SCHEMBL30251598 0.82 TSHR (0.64) NPC1RAB9ASMN1; SMN2ALDH1A1KMT2A
SCHEMBL866718 0.82 TSHR (0.64) NPC1RAB9ASMN1; SMN2ALDH1A1KMT2A
SCHEMBL8993085 0.82 ADRB3 (0.50) NPC1RAB9ASMN1; SMN2MAPK1ALDH1A1
SCHEMBL2093768 0.82 AOC3 (0.59) NPC1RAB9AMAPK1ALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed