SCHEMBL8993230

SCHEMBL8993230

Cc1ccc2c(c1N=C1N=CCO1)CCC(C)C2

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.34
CYP2A13 Q16696 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TSHR P16473 1/20 0.34
TRPV1 Q8NER1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8993327 0.90 CYP2A6 (0.31) CYP2A6CYP2A13ALDH1A1TSHR
SCHEMBL8993415 0.76 CYP2A6 (0.31) CYP2A6CYP2A13ALDH1A1TSHR
SCHEMBL8625418 0.73 CYP2A6 (0.35) CYP2A6CYP2A13ALDH1A1TSHR
SCHEMBL12511860 0.65 ALDH1A1 (0.42) CYP2A6CYP2A13ALDH1A1TSHR
SCHEMBL12433438 0.65 CYP2A6 (0.42) CYP2A6CYP2A13ALDH1A1TSHRTRPV1
SCHEMBL24718000 0.65 ALDH1A1 (0.42) CYP2A6CYP2A13ALDH1A1TSHR
SCHEMBL19032997 0.65 ALDH1A1 (0.42) CYP2A6CYP2A13ALDH1A1TSHR
SCHEMBL23510011 0.65 ALDH1A1 (0.42) CYP2A6CYP2A13ALDH1A1TSHR
SCHEMBL19999344 0.63 ADRA2A (0.44) CYP2A6CYP2A13ALDH1A1TSHR
SCHEMBL8622879 0.62 CYP2A6 (0.32) CYP2A6CYP2A13ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0724439-A1 USE OF 2-(2-ALKYLPHENYLAMINO)-OXAZOLINES, -THIAZOLINES AND -IMIDAZOLINES AS ALPHA 2 ADRENERGIC AGENTS Allergan (US) 1996-08-07 EP disclosed
WO-1995011021-A1 USE OF 2-(2-ALKYLPHENYLAMINO)-OXAZOLINES, -THIAZOLINES AND -IMIDAZOLINES AS ALPHA 2 ADRENERGIC AGENTS ALLERGAN (US) 1995-04-27 WO disclosed