SCHEMBL8993378

SCHEMBL8993378

Cc1ccc(S(=O)(=O)CC2=CCCC2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 2/20 0.40
TSHR P16473 1/20 0.40
ESR1 P03372 1/20 0.40
POLB P06746 1/20 0.40
NR4A1 P22736 1/20 0.40
APEX1 P27695 1/20 0.40
RECQL P46063 1/20 0.40
DUSP3 P51452 1/20 0.40
PTPN5 P54829 1/20 0.40
PTPN11 Q06124 1/20 0.40
ESR2 Q92731 1/20 0.40
CTDSP1 Q9GZU7 1/20 0.40
MCHR1 Q99705 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22305967 0.80 ALDH1A1 (0.53) ALDH1A1CYP3A4CYP2C9CYP2C19MEN1
SCHEMBL7070454 0.78 KMT2A (0.38) ALDH1A1MEN1KMT2AHSD17B10TDP1
SCHEMBL7070187 0.75 MEN1 (0.42) ALDH1A1CYP2C9CYP2C19MEN1KMT2A
SCHEMBL19318751 0.70 GAA (0.54) ALDH1A1MEN1KMT2APOLBGAA
SCHEMBL9820117 0.70 ALDH1A1 (0.59) ALDH1A1CYP3A4CYP2C9CYP2C19MEN1
SCHEMBL16221401 0.70 TDP1 (0.76) ALDH1A1MEN1KMT2AHSD17B10TDP1
SCHEMBL21494752 0.69 KMT2A (0.47) ALDH1A1MEN1KMT2ATDP1POLB
SCHEMBL7148200 0.69 ALDH1A1 (0.57) ALDH1A1CYP3A4CYP2C9CYP2C19MEN1
SCHEMBL25654792 0.69 ALDH1A1 (0.41) ALDH1A1MEN1KMT2ATDP1
SCHEMBL25654790 0.68 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0724566-A1 1,2-DIARYLCYCLOPENTENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-08-07 EP disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
WO-1995011883-A1 1,2-DIARYLCYCLOPENTENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-05-04 WO disclosed