SCHEMBL8993386

SCHEMBL8993386

CC1SC2=C(c3ccc(F)cc31)N(c1ccc(S(N)(=O)=O)cc1)NC2(C(=O)O)C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.33
PTGS1 P23219 6/20 0.33
CHRNA7 P36544 3/20 0.33
CA1 P00915 3/20 0.33
CA2 P00918 3/20 0.33
CA9 Q16790 2/20 0.33
CA4 P22748 2/20 0.33
CA12 O43570 1/20 0.32
CA7 P43166 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8933875 0.81 PTGS2 (0.47) PTGS2PTGS1CA1CA2CA9
SCHEMBL8993413 0.67 PTGS2 (0.47) PTGS2PTGS1CHRNA7CA1CA2
SCHEMBL8828054 0.65 PTGS2 (0.47) PTGS2PTGS1CHRNA7CA1CA2
Trifluoroacetic Acid SCHEMBL27865608 0.57 CA2 (0.59) PTGS2PTGS1CA1CA2CA9
SCHEMBL6352339 0.55 PTGS2 (0.81) PTGS2PTGS1CA1CA2CA9
SCHEMBL8688866 0.55 PTGS2 (0.46) PTGS2PTGS1CA1CA2CA9
SCHEMBL3245730 0.55 PTGS2 (0.77) PTGS2PTGS1
SCHEMBL5857453 0.54 PTGS2 (0.46) PTGS2PTGS1CA1CA2CA9
SCHEMBL8689162 0.53 PTGS2 (0.46) PTGS2PTGS1CA1CA2CA9
SCHEMBL7216763 0.53 CHRNA7 (0.62) PTGS2PTGS1CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5547975-A ANTIARTHRIC AGENTS, ANALGESICS AND ANTIPYRETICS; INHIBITORS OF CYCLOOXYGENASE II; SIDE EFFECT REDUCTION G.D. SEARLE & CO. 1996-08-20 US disclosed