SCHEMBL8996040

SCHEMBL8996040

Cn1ncnc1C(=O)NCCN

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.42
CYP1A2 P05177 2/20 0.39
TSHR P16473 1/20 0.39
NFKB1 P19838 1/20 0.39
KDM4E B2RXH2 1/20 0.38
PMP22 Q01453 2/20 0.38
MEN1 O00255 1/20 0.38
BLM P54132 1/20 0.38
KMT2A Q03164 1/20 0.38
JAK2 O60674 1/20 0.37
FLT3 P36888 1/20 0.37
SYK P43405 1/20 0.37
TERT O14746 2/20 0.36
CYP3A4 P08684 1/20 0.35
THPO P40225 1/20 0.35
AKT3 Q9Y243 1/20 0.35
LMNA P02545 1/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8950151 0.80 MAOB (0.39) MAOBCYP1A2TSHRNFKB1KDM4E
SCHEMBL8996043 0.71 KDM4E (0.42) TSHRKDM4ECA12CA1CA2
SCHEMBL12496155 0.71
SCHEMBL510655 0.67 GAA (0.33) TSHRKDM4EMEN1KMT2ALMNA
SCHEMBL8954913 0.66 BRD4 (0.40) KDM4EKMT2ALMNARAB9A
SCHEMBL25458163 0.65 KDM4E (0.33) TSHRKDM4EBLMKMT2ALMNA
SCHEMBL10897204 0.65 PREP (0.45) MAOBCYP1A2TSHRNFKB1KDM4E
SCHEMBL20369065 0.65 MAOB (0.45) MAOBCYP1A2TSHRNFKB1PMP22
SCHEMBL28224466 0.65 GAA (0.52) MAOBCYP1A2TSHRNFKB1MEN1
SCHEMBL1655108 0.64 HCAR2 (0.56) MAOBCYP1A2TSHRNFKB1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188085-B2 Antifungal agents MERCK SHARP & DOHME CORP. (US) 2012-05-29 US disclosed
US-20100113439-A1 Antifungal agents MERCK & CO., INC. (US) 2010-05-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100113439-A1 Antifungal agents GMDS, GBA3, UGGT1 MAOB 2163/4885CYP1A2 623/4885TSHR 4815/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.