SCHEMBL8996336

SCHEMBL8996336

COc1cc(-c2nc3ccccc3[nH]2)cc2c1C(=O)c1c(O)cccc1C2=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
AMY1A P0DUB6 5/20 0.47
KMT2A Q03164 3/20 0.46
DHODH Q02127 1/20 0.46
CYP1A1 P04798 2/20 0.46
CYP1B1 Q16678 2/20 0.46
CYP1A2 P05177 1/20 0.46
CDK4 P11802 1/20 0.46
CCNA2 P20248 1/20 0.46
CCND1 P24385 1/20 0.46
CDK2 P24941 1/20 0.46
CCND3 P30281 1/20 0.46
MEN1 O00255 2/20 0.45
F7 P08709 1/20 0.45
EGFR P00533 1/20 0.44
PIM1 P11309 1/20 0.44
USP2 O75604 1/20 0.44
CASP3 P42574 1/20 0.44
ATM Q13315 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8996330 0.92 AMY1A (0.54) NPC1RAB9AAMY1AKMT2ADHODH
SCHEMBL8996325 0.88 F7 (0.51) NPC1RAB9AKMT2AMEN1F7
SCHEMBL8996340 0.82 KDM4E (0.54) NPC1RAB9AAMY1AKMT2AMEN1
Hydrochloric Acid SCHEMBL8996365 0.81 KDM4E (0.53) NPC1RAB9AAMY1AKMT2AMEN1
SCHEMBL8996422 0.79 KMT2A (0.50) NPC1RAB9AAMY1AKMT2AMEN1
SCHEMBL24140790 0.76 AMY1A (0.62) NPC1RAB9AAMY1AKMT2ACYP1A1
SCHEMBL7395130 0.76 AMY1A (0.69) NPC1RAB9AAMY1AKMT2AUSP2
SCHEMBL31429770 0.75 AMY1A (0.62) NPC1RAB9AAMY1AKMT2AMEN1
SCHEMBL15456540 0.74 CYP1A1 (0.69) NPC1RAB9AAMY1AKMT2ACYP1A1
SCHEMBL8930315 0.72 MAPT (0.73) KMT2AMEN1EGFRPIM1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5480873-A ARTHRITIS LILLY INDUSTRIES LIMITED (GB) 1996-01-02 US disclosed
EP-0570091-A1 Anthraquinone derivatives, process for their preparation and their use as medicaments LILLY INDUSTRIES LIMITED (GB) 1993-11-18 EP disclosed