SCHEMBL8997158

SCHEMBL8997158

Nc1nc(O)c2c(n1)NCC2CCc1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc1

nearest known ligand 0.68

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ATIC P31939 2/20 0.61
GART P22102 6/20 0.59
DHFR P00374 3/20 0.52
TYMS P04818 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12521635 1.00 ATIC (0.61) ATICGARTDHFRTYMS
SCHEMBL9227067 0.97 ATIC (0.58) ATICGARTDHFRTYMS
SCHEMBL8997205 0.95 GART (0.60) ATICGARTDHFRTYMS
SCHEMBL9223778 0.92 GART (0.57) ATICGARTDHFR
SCHEMBL9227075 0.90 ATIC (0.51) ATICGARTDHFRTYMS
SCHEMBL9432057 0.87 GART (0.60) ATICGARTDHFRTYMS
SCHEMBL8997257 0.87 GART (0.61) ATICGARTDHFR
Lometrexol SCHEMBL12022771 0.85 GART (0.75) ATICGARTDHFRTYMS
Lometrexol SCHEMBL9045915 0.85 GART (0.75) ATICGARTDHFRTYMS
SCHEMBL13575748 0.85 ATIC (0.79) ATICGARTDHFRTYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997838-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-03-05 US claimed
EP-0334636-B1 Pyrrolopyrimidine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-10-23 EP disclosed
US-5539113-A ANTITUMOR AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-07-23 US disclosed
US-5296600-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-22 US disclosed
US-5106974-A Antitumor and -carcinogenic agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-04-21 US disclosed
US-4997838-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-03-05 US disclosed