SCHEMBL8997205

SCHEMBL8997205

Nc1nc(O)c2c(n1)NCC2CCCc1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc1

nearest known ligand 0.65

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GART P22102 7/20 0.60
ATIC P31939 3/20 0.57
DHFR P00374 4/20 0.54
TYMS P04818 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9223778 0.97 GART (0.57) GARTATICDHFR
SCHEMBL12521635 0.95 ATIC (0.61) GARTATICDHFRTYMS
SCHEMBL8997158 0.95 ATIC (0.61) GARTATICDHFRTYMS
SCHEMBL9432057 0.92 GART (0.60) GARTATICDHFRTYMS
SCHEMBL8997257 0.92 GART (0.61) GARTATICDHFR
SCHEMBL9227067 0.92 ATIC (0.58) GARTATICDHFRTYMS
SCHEMBL9223785 0.90 GART (0.51) GARTATICDHFR
SCHEMBL9446110 0.89 ATIC (0.69) GARTATICDHFRTYMS
SCHEMBL9048275 0.86 GART (0.69) GARTATICDHFR
SCHEMBL9439358 0.86 GART (0.58) GARTATIC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997838-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-03-05 US claimed
EP-0334636-B1 Pyrrolopyrimidine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-10-23 EP disclosed
US-5539113-A ANTITUMOR AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-07-23 US disclosed
US-5496946-A Production of pyrrolopyrimidines and intermediates therefor TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-03-05 US disclosed
US-5349064-A Production of pyrrolopyrimidines TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-09-20 US disclosed
US-5296600-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-22 US disclosed
US-5106974-A Antitumor and -carcinogenic agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-04-21 US disclosed
US-4997838-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-03-05 US disclosed
EP-0402903-A1 Production of pyrrolopyrimidines and intermediates therefor Takeda Chemical Industries, Ltd. (JP) 1990-12-19 EP disclosed
EP-0334636-A2 Pyrrolopyrimidine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-09-27 EP disclosed