SCHEMBL8997212

SCHEMBL8997212

COC(=O)c1ccc(CCCC2CN=C3NC(N)=NC(O)=C32)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4A11 Q02928 2/20 0.42
CYP4F2 P78329 1/20 0.41
LOXL2 Q9Y4K0 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
MAPT P10636 1/20 0.35
TP53 P04637 2/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
HPGD P15428 1/20 0.35
ALOX15 P16050 1/20 0.35
ALOX12 P18054 1/20 0.35
CYP2C19 P33261 1/20 0.35
CKS1B P61024 1/20 0.35
SKP2 Q13309 1/20 0.35
HIF1A Q16665 1/20 0.35
HSD17B10 Q99714 1/20 0.35
DHODH Q02127 1/20 0.34
TLR8 Q9NR97 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8997438 0.82 SIRT2 (0.36) CYP4A11CYP4F2ALOX15CA1CA2
SCHEMBL8997209 0.68 CYP4A11 (0.43) CYP4A11CYP4F2LOXL2TP53ALDH1A1
SCHEMBL12176878 0.65 CYP4A11 (0.70) CYP4A11CYP4F2LOXL2MAPTTP53
SCHEMBL19922842 0.65 CYP4A11 (0.60) CYP4A11CYP4F2LOXL2TP53ALDH1A1
SCHEMBL7505320 0.65 CYP4A11 (0.60) CYP4A11CYP4F2LOXL2SMN1; SMN2MAPT
SCHEMBL7987096 0.65 CYP4A11 (0.56) CYP4A11CYP4F2LOXL2TP53ALDH1A1
Hydrochloric Acid SCHEMBL19585552 0.64 CYP4A11 (0.55) CYP4A11CYP4F2LOXL2HRH1
SCHEMBL5733406 0.64 CYP4A11 (0.72) CYP4A11CYP4F2LOXL2MAPTTP53
SCHEMBL70185 0.63 CYP4A11 (0.75) CYP4A11CYP4F2LOXL2SMN1; SMN2MAPT
SCHEMBL28281244 0.62 CYP4A11 (0.73) CYP4A11CYP4F2LOXL2MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0334636-B1 Pyrrolopyrimidine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-10-23 EP disclosed
US-5539113-A ANTITUMOR AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-07-23 US disclosed
US-5296600-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-22 US disclosed
US-5106974-A Antitumor and -carcinogenic agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-04-21 US disclosed
US-4997838-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-03-05 US disclosed
EP-0334636-A2 Pyrrolopyrimidine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-09-27 EP disclosed