SCHEMBL8997380

SCHEMBL8997380

COC(=O)C(I)CCCc1ccc(C(=O)OC(C)(C)C)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4A11 Q02928 3/20 0.47
CYP4F2 P78329 2/20 0.46
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA12 O43570 1/20 0.37
CA9 Q16790 1/20 0.37
CA14 Q9ULX7 1/20 0.37
LOXL2 Q9Y4K0 1/20 0.37
MMP3 P08254 2/20 0.37
MMP1 P03956 1/20 0.37
MMP9 P14780 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.36
SIRT1 Q96EB6 1/20 0.36
NPC1 O15118 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36
SMO Q99835 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9446036 0.82 CYP4A11 (0.45) CYP4A11CYP4F2CA1CA2CA12
SCHEMBL8997190 0.81 CYP4A11 (0.43) CYP4A11CYP4F2CA1CA2CA12
SCHEMBL8568070 0.80 CYP4A11 (0.45) CYP4A11CYP4F2CA1CA2CA12
SCHEMBL7428977 0.78 CYP4A11 (0.45) CYP4A11CYP4F2CA1CA2CA12
SCHEMBL31688879 0.78 CYP4A11 (0.49) CYP4A11CYP4F2CA1CA2CA12
SCHEMBL8562574 0.78 CYP4A11 (0.49) CYP4A11CYP4F2CA1CA2CA12
SCHEMBL9439645 0.77 HPGD (0.41) TAS1R3TAS1R1HDAC1HDAC6ALDH1A1
SCHEMBL6209198 0.76 CYP4A11 (0.50) CYP4A11CYP4F2CA1CA2CA12
SCHEMBL7855043 0.76 CYP4A11 (0.68) CYP4A11CYP4F2CA1CA2CA12
SCHEMBL9446097 0.76 CYP4A11 (0.46) CYP4A11CYP4F2CA1CA2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0334636-B1 Pyrrolopyrimidine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-10-23 EP disclosed
US-5539113-A ANTITUMOR AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-07-23 US disclosed
US-5296600-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-22 US disclosed
US-5106974-A Antitumor and -carcinogenic agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-04-21 US disclosed
US-4997838-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-03-05 US disclosed
EP-0334636-A2 Pyrrolopyrimidine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-09-27 EP disclosed