SCHEMBL9439645

SCHEMBL9439645

COC(=O)C(I)CCCc1ccc(C(=O)OC(C)(C)C)s1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.41
NPSR1 Q6W5P4 2/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
ATM Q13315 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
LMNA P02545 2/20 0.35
ALDH1A1 P00352 1/20 0.35
PRNP P04156 1/20 0.35
RECQL P46063 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
POLB P06746 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
MRGPRX4 Q96LA9 1/20 0.33
PTGER4 P35408 3/20 0.33
TRPV1 Q8NER1 1/20 0.32
HDAC3 O15379 1/20 0.31
HDAC4 P56524 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5050275 0.79 HPGD (0.42) HPGDNPSR1TSHRMAPK1ATM
Hydrochloric Acid SCHEMBL5724631 0.78 HPGD (0.41) HPGDNPSR1TSHRMAPK1ATM
SCHEMBL8570240 0.78 HPGD (0.43) HPGDNPSR1TSHRMAPK1ATM
Hydrochloric Acid SCHEMBL2413233 0.78 HPGD (0.40) HPGDNPSR1TSHRMAPK1ATM
SCHEMBL9439542 0.78 HPGD (0.67) HPGDNPSR1TSHRMAPK1ATM
SCHEMBL8564545 0.77 HPGD (0.45) HPGDNPSR1TSHRMAPK1ATM
SCHEMBL21199747 0.77 POLB (0.46) HPGDNPSR1TSHRMAPK1ATM
SCHEMBL8982459 0.77 HPGD (0.45) HPGDNPSR1TSHRMAPK1ATM
SCHEMBL8997380 0.77 CYP4A11 (0.47) HPGDL3MBTL1ALDH1A1HDAC1HDAC6
SCHEMBL4197199 0.77 HPGD (0.70) HPGDNPSR1TSHRMAPK1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354754-A Antitumor and -carcinogenic agents; treating human epidermoid carcinoma KB TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-10-11 US disclosed
EP-0418924-A2 Pyrrolopyrimidines, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-03-27 EP disclosed