SCHEMBL8998726

SCHEMBL8998726

CC(C)N1CC=CC(N)=C1N1CCN(C(=O)c2cc3cc(NS(C)(=O)=O)ccc3[nH]2)CC1

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.57
ADORA3 P0DMS8 1/20 0.57
CHRM1 P11229 1/20 0.57
MAOA P21397 1/20 0.57
TBXA2R P21731 1/20 0.57
OPRM1 P35372 1/20 0.57
MDH1 P40925 1/20 0.57
KCNH2 Q12809 1/20 0.57
ABCG2 Q9UNQ0 1/20 0.57
HRH3 Q9Y5N1 4/20 0.45
MMP2 P08253 1/20 0.43
MMP13 P45452 1/20 0.43
HRH4 Q9H3N8 8/20 0.43
HRH1 P35367 1/20 0.41
SYK P43405 2/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27672437 0.75 HRH4 (0.65) ADRA2AADORA3CHRM1MAOATBXA2R
SCHEMBL14571138 0.73 ADRA2A (0.59) ADRA2AADORA3CHRM1MAOATBXA2R
Delavirdine SCHEMBL29602259 0.72 ADRA2A (1.00) ADRA2AADORA3CHRM1MAOATBXA2R
Delavirdine SCHEMBL29714124 0.72 ADRA2A (1.00) ADRA2AADORA3CHRM1MAOATBXA2R
Delavirdine SCHEMBL30803764 0.72 ADRA2A (1.00) ADRA2AADORA3CHRM1MAOATBXA2R
Delavirdine SCHEMBL34420 0.72 ADRA2A (1.00) ADRA2AADORA3CHRM1MAOATBXA2R
Delavirdine SCHEMBL40522 0.72 ADRA2A (0.98) ADRA2AADORA3CHRM1MAOATBXA2R
Delavirdine SCHEMBL29585604 0.72 ADRA2A (0.98) ADRA2AADORA3CHRM1MAOATBXA2R
Delavirdine SCHEMBL3221265 0.72 ADRA2A (0.98) ADRA2AADORA3CHRM1MAOATBXA2R
Delavirdine SCHEMBL28170537 0.72 ADRA2A (0.98) ADRA2AADORA3CHRM1MAOATBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729948-A1 The production of 3-alkylamino-2-piperazinylpyridines THE UPJOHN COMPANY (US) 1996-09-04 EP disclosed