SCHEMBL27672437

SCHEMBL27672437

CS(=O)(=O)Nc1ccc2[nH]c(C(=O)N3CCNCC3)cc2c1

nearest known ligand 0.66

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 12/20 0.65
ADRA2A P08913 1/20 0.58
ADORA3 P0DMS8 1/20 0.58
CHRM1 P11229 1/20 0.58
MAOA P21397 1/20 0.58
TBXA2R P21731 1/20 0.58
OPRM1 P35372 1/20 0.58
MDH1 P40925 1/20 0.58
KCNH2 Q12809 1/20 0.58
ABCG2 Q9UNQ0 1/20 0.58
HRH3 Q9Y5N1 5/20 0.58
MMP2 P08253 1/20 0.57
MMP13 P45452 1/20 0.57
SYK P43405 1/20 0.53
HRH1 P35367 1/20 0.51
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17938665 0.79 NPC1 (0.78) HRH4HRH3NPC1RAB9A
SCHEMBL6130879 0.79 HRH4 (1.00) HRH4HRH3HRH1RAB9A
SCHEMBL8406457 0.79 MMP13 (0.68) ADRA2AADORA3CHRM1MAOATBXA2R
SCHEMBL12862876 0.79 MMP13 (0.68) ADRA2AADORA3CHRM1MAOATBXA2R
SCHEMBL27672435 0.78 HRH4 (0.60) HRH4HRH3SYKHRH1NPC1
SCHEMBL14899883 0.77 HRH4 (0.73) HRH4HRH3HRH1NPC1RAB9A
SCHEMBL8781424 0.76 SIGMAR1 (0.55) NPC1RAB9A
SCHEMBL22091300 0.76 HRH4 (0.60) HRH4HRH3SYK
SCHEMBL8998726 0.75 ADRA2A (0.57) HRH4ADRA2AADORA3CHRM1MAOA
Delavirdine SCHEMBL34420 0.75 ADRA2A (1.00) ADRA2AADORA3CHRM1MAOATBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102304150-A Phospho-indoles as HIV inhibitors IDENIX PHARMACEUTICALS INC (US) 2012-01-04 CN disclosed
CN-100343268-C Beta-2 '-or 3' -halonucleosides PHARMASSET LTD (BB) 2007-10-17 CN disclosed