SCHEMBL8998855

SCHEMBL8998855

CONC(=O)CCc1c[nH]c2ccccc12

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.72
ALDH1A1 P00352 2/20 0.72
GAA P10253 1/20 0.72
HPGD P15428 2/20 0.62
HTT P42858 1/20 0.62
RECQL P46063 1/20 0.62
MEN1 O00255 4/20 0.60
KMT2A Q03164 4/20 0.60
KDM4E B2RXH2 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
FAAH O00519 1/20 0.57
GFER P55789 1/20 0.57
LMNA P02545 1/20 0.57
CYP1A2 P05177 1/20 0.57
PKM P14618 1/20 0.57
TSHR P16473 1/20 0.57
CYP2C19 P33261 1/20 0.57
BLM P54132 1/20 0.57
EGFR P00533 1/20 0.56
SRC P12931 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29634969 1.00 MAPT (0.72) MAPTALDH1A1GAAHPGDHTT
SCHEMBL6275395 0.84 ALDH1A1 (0.74) MAPTALDH1A1GAAHPGDHTT
Methyl 3-(3-Indolylmethyl)Propanoate SCHEMBL290808 0.84 MAPT (0.71) MAPTALDH1A1GAAHPGDHTT
SCHEMBL393877 0.84 MAPT (1.00) MAPTALDH1A1GAAHPGDHTT
SCHEMBL12371556 0.84 MAPT (0.78) MAPTALDH1A1GAAHPGDHTT
SCHEMBL21178436 0.83 MAPT (0.64) MAPTALDH1A1GAAHPGDHTT
SCHEMBL1520411 0.82 MAPT (0.76) MAPTALDH1A1GAAHPGDHTT
SCHEMBL13973308 0.82 MAPT (0.74) MAPTALDH1A1GAAHPGDHTT
SCHEMBL30674423 0.81 MEN1 (0.65) MAPTALDH1A1GAAHPGDHTT
SCHEMBL26708909 0.81 MEN1 (0.65) MAPTALDH1A1GAAHPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5556874-A ENZYME INHIBITORS AS ANTICARCINOGENIC AGENTS WARNER LAMBERT COMPANY (US) 1996-09-17 US disclosed
US-5464861-A Anticarcinogenic agents WARNER-LAMBERT (US) 1995-11-07 US disclosed
EP-0654024-A1 2-THIOINDOLES (SELENOINDOLES) AND RELATED DISULFIDES (SELENIDES) WHICH INHIBIT PROTEIN TYROSINE KINASES AND WHICH HAVE ANTITUMOR PROPERTIES WARNER-LAMBERT COMPANY (US) 1995-05-24 EP disclosed
WO-1994003427-A1 2-THIOINDOLES (SELENOINDOLES) AND RELATED DISULFIDES (SELENIDES) WHICH INHIBIT PROTEIN TYROSINE KINASES AND WHICH HAVE ANTITUMOR PROPERTIES WARNER-LAMBERT COMPANY (US) 1994-02-17 WO disclosed