SCHEMBL8998871

SCHEMBL8998871

CC(=O)Oc1ccc2c(c1)N(C)C(=S)C2

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.41
CA2 P00918 1/20 0.41
CA5A P35218 1/20 0.41
POLB P06746 3/20 0.39
HTT P42858 1/20 0.39
KDM4E B2RXH2 2/20 0.39
LMNA P02545 2/20 0.39
CYP3A4 P08684 1/20 0.38
GLA P06280 2/20 0.38
ACHE P22303 1/20 0.38
OPRD1 P41143 1/20 0.37
MAPT P10636 2/20 0.36
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CA12 O43570 1/20 0.36
GAA P10253 1/20 0.36
CA9 Q16790 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
PKM P14618 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8998941 0.88 MAPT (0.39) OPRM1CA2CA5APOLBHTT
SCHEMBL8998821 0.84 GLA (0.45) OPRM1CA2CA5APOLBHTT
SCHEMBL10828319 0.73 NOTUM (0.56) OPRM1CA2CA5APOLBKDM4E
SCHEMBL8999438 0.72 GAA (0.48) POLBLMNAGLAMAPTALDH1A1
SCHEMBL6536539 0.71 MAPT (0.53) CA2CA5APOLBKDM4ELMNA
SCHEMBL8999088 0.71 ALDH1A1 (0.37) CYP3A4MAPTALDH1A1CA12GAA
SCHEMBL8999027 0.69 SRD5A1 (0.40) OPRM1CA2POLBKDM4ELMNA
SCHEMBL8998850 0.68 MAPK1 (0.39) POLBKDM4ELMNAACHEMAPT
SCHEMBL8999080 0.68 MAPK1 (0.42) POLBKDM4ELMNAACHEMAPT
SCHEMBL8998856 0.67 DRD1 (0.47) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5556874-A ENZYME INHIBITORS AS ANTICARCINOGENIC AGENTS WARNER LAMBERT COMPANY (US) 1996-09-17 US disclosed
US-5464861-A Anticarcinogenic agents WARNER-LAMBERT (US) 1995-11-07 US disclosed
EP-0654024-A1 2-THIOINDOLES (SELENOINDOLES) AND RELATED DISULFIDES (SELENIDES) WHICH INHIBIT PROTEIN TYROSINE KINASES AND WHICH HAVE ANTITUMOR PROPERTIES WARNER-LAMBERT COMPANY (US) 1995-05-24 EP disclosed
WO-1994003427-A1 2-THIOINDOLES (SELENOINDOLES) AND RELATED DISULFIDES (SELENIDES) WHICH INHIBIT PROTEIN TYROSINE KINASES AND WHICH HAVE ANTITUMOR PROPERTIES WARNER-LAMBERT COMPANY (US) 1994-02-17 WO disclosed