SCHEMBL8999230

SCHEMBL8999230

N#C/C(Br)=C(\c1ccccc1)c1ccc(CBr)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.53
CES1 P23141 1/20 0.53
ALDH1A1 P00352 2/20 0.43
TRPA1 O75762 1/20 0.43
TSHR P16473 1/20 0.43
CYP19A1 P11511 2/20 0.39
SNCA P37840 2/20 0.39
CYP1A1 P04798 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP1B1 Q16678 2/20 0.36
ESR1 P03372 4/20 0.34
PTPN1 P18031 1/20 0.33
GSK3B P49841 1/20 0.33
ESR2 Q92731 1/20 0.32
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8999238 1.00 CES2 (0.53) CES2CES1ALDH1A1TRPA1TSHR
SCHEMBL14756543 0.81 CES2 (0.69) CES2CES1ALDH1A1TRPA1TSHR
SCHEMBL68718 0.81 CES2 (0.69) CES2CES1ALDH1A1TRPA1TSHR
SCHEMBL68719 0.81 CES2 (0.69) CES2CES1ALDH1A1TRPA1TSHR
SCHEMBL8999241 0.79 CES2 (0.49) CES2CES1ALDH1A1TRPA1TSHR
SCHEMBL8999233 0.79 CES2 (0.49) CES2CES1ALDH1A1TRPA1TSHR
SCHEMBL8998998 0.79 CES2 (0.47) CES2CES1ALDH1A1TSHRCYP19A1
SCHEMBL8998995 0.79 CES2 (0.47) CES2CES1ALDH1A1TSHRCYP19A1
SCHEMBL21241545 0.73 CES2 (0.58) CES2CES1ALDH1A1TRPA1TSHR
Benzyl Bromide SCHEMBL28292772 0.72 ALDH1A1 (0.74) CES2CES1ALDH1A1TRPA1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5554624-A CONGESTIVE HEART FAILURE; HYPOTENSIVE AGENTS J. URIACH & CIA. (ES) 1996-09-10 US disclosed
EP-0669333-A1 New imidazopyridine derivatives as angiotensin II antagonists J. URIACH & CIA. S.A. (ES) 1995-08-30 EP disclosed