SCHEMBL8999345

SCHEMBL8999345

O=C(O)C=C(c1ccccc1)c1ccccc1CBr

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.40
GSK3B P49841 1/20 0.40
CES1 P23141 2/20 0.40
CES2 O00748 1/20 0.40
PDPK1 O15530 4/20 0.38
KDM4E B2RXH2 2/20 0.37
CYP3A4 P08684 2/20 0.37
MAPT P10636 2/20 0.37
HPGD P15428 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
TSHR P16473 1/20 0.36
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
NFE2L2 Q16236 1/20 0.35
AKR1C3 P42330 1/20 0.35
FOLH1 Q04609 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
NCOR2 Q9Y618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7826090 0.80 PDPK1 (0.44) PTPN1GSK3BCES1CES2PDPK1
SCHEMBL8948923 0.78 HTT (0.40) KDM4EHPGDAKR1C3FOLH1ALOX15
SCHEMBL3093625 0.77 AKR1C3 (0.55) PTPN1GSK3BCES1CES2MAPT
SCHEMBL8999341 0.76 CES2 (0.65) PTPN1GSK3BCES1CES2PDPK1
SCHEMBL7955212 0.75 ALDH1A1 (0.38) CES1CES2PDPK1KDM4ETSHR
SCHEMBL27296890 0.75 PDE4A (0.45) PTPN1GSK3BCES1CES2
SCHEMBL63954 0.75 CES1 (0.50) CES1CES2KDM4ECYP3A4MAPT
SCHEMBL3978126 0.75 CES2 (0.58) PTPN1GSK3BCES1CES2MAPT
SCHEMBL8948909 0.74 ALDH1A1 (0.43) KDM4EHPGDSMN1; SMN2TSHRKMT2A
SCHEMBL8948905 0.74 ALDH1A1 (0.43) KDM4EHPGDSMN1; SMN2TSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5554624-A CONGESTIVE HEART FAILURE; HYPOTENSIVE AGENTS J. URIACH & CIA. (ES) 1996-09-10 US disclosed
EP-0669333-A1 New imidazopyridine derivatives as angiotensin II antagonists J. URIACH & CIA. S.A. (ES) 1995-08-30 EP disclosed