SCHEMBL9001820

SCHEMBL9001820

CC(CCn1ccc2nc(N)[nH]c(=O)c21)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)o1

nearest known ligand 0.68

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ATIC P31939 15/20 0.68
SHMT1 P34896 14/20 0.68
SHMT2 P34897 14/20 0.68
GART P22102 11/20 0.67
DHFR P00374 3/20 0.54
TYMS P04818 1/20 0.54
FOLR2 P14207 1/20 0.48
FOLR1 P15328 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9001842 0.93 ATIC (0.64) ATICSHMT1SHMT2GARTDHFR
SCHEMBL9001757 0.91 ATIC (0.66) ATICSHMT1SHMT2GARTDHFR
SCHEMBL9001815 0.88 ATIC (0.52) ATICSHMT1SHMT2GARTDHFR
SCHEMBL9001806 0.87 ATIC (0.72) ATICSHMT1SHMT2GARTDHFR
SCHEMBL9001772 0.86 ATIC (0.63) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8571085 0.86 ATIC (0.49) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8571094 0.86 ATIC (0.49) ATICSHMT1SHMT2GARTDHFR
SCHEMBL9001756 0.85 ATIC (0.78) ATICSHMT1SHMT2GARTDHFR
SCHEMBL9001850 0.85 ATIC (0.75) ATICSHMT1SHMT2GARTDHFR
SCHEMBL9001790 0.84 ATIC (0.73) ATICSHMT1SHMT2GARTDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed