SCHEMBL9001850

SCHEMBL9001850

CC(CCn1ccc2nc(N)[nH]c(=O)c21)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc1

nearest known ligand 0.75

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ATIC P31939 15/20 0.75
SHMT1 P34896 14/20 0.75
SHMT2 P34897 14/20 0.75
GART P22102 13/20 0.75
DHFR P00374 2/20 0.59
TYMS P04818 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9001846 0.92 ATIC (0.71) ATICSHMT1SHMT2GARTDHFR
SCHEMBL9001755 0.90 ATIC (0.73) ATICSHMT1SHMT2GARTDHFR
SCHEMBL9001843 0.87 GART (0.57) ATICSHMT1SHMT2GARTDHFR
SCHEMBL9001784 0.87 ATIC (0.90) ATICSHMT1SHMT2GARTDHFR
SCHEMBL9001780 0.86 ATIC (0.77) ATICSHMT1SHMT2GARTDHFR
SCHEMBL9001862 0.86 ATIC (0.69) ATICSHMT1SHMT2GARTDHFR
SCHEMBL20854920 0.86 ATIC (1.00) ATICSHMT1SHMT2GARTDHFR
SCHEMBL9001800 0.86 ATIC (1.00) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8564656 0.85 DHFR (0.56) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8564651 0.85 DHFR (0.56) ATICSHMT1SHMT2GARTDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed