SCHEMBL9001891

SCHEMBL9001891

NC[CH]C(=O)OCc1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.61
LMNA P02545 2/20 0.57
ALDH1A1 P00352 5/20 0.53
CA12 O43570 3/20 0.53
CA9 Q16790 3/20 0.53
AKR1B10 O60218 2/20 0.53
AKR1B1 P15121 2/20 0.53
CA4 P22748 1/20 0.53
CA6 P23280 1/20 0.53
CA5A P35218 1/20 0.53
CA7 P43166 1/20 0.53
CA14 Q9ULX7 1/20 0.53
CA5B Q9Y2D0 1/20 0.53
TDP1 Q9NUW8 2/20 0.52
MAPK1 P28482 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
SLC6A2 P23975 1/20 0.52
SLC6A3 Q01959 1/20 0.52
KMT2A Q03164 1/20 0.52
TTR P02766 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3094482 0.86 HCAR2 (0.57) HCAR2LMNAALDH1A1CA12CA9
SCHEMBL4065633 0.83 HCAR2 (0.62) HCAR2LMNAALDH1A1CA12CA9
SCHEMBL7719568 0.82 HCAR2 (0.67) HCAR2LMNAALDH1A1CA12CA9
SCHEMBL14675315 0.82 HCAR2 (0.53) HCAR2LMNAALDH1A1CA12CA9
SCHEMBL9650418 0.81 HCAR2 (0.61) HCAR2LMNAALDH1A1CA12CA9
SCHEMBL6133091 0.81 HCAR2 (0.61) HCAR2LMNAALDH1A1CA12CA9
SCHEMBL14940404 0.81 HCAR2 (0.65) HCAR2LMNAALDH1A1CA12CA9
SCHEMBL337503 0.80 HCAR2 (0.89) HCAR2LMNAALDH1A1CA12CA9
SCHEMBL9395526 0.80 HCAR2 (0.69) HCAR2LMNAALDH1A1CA12CA9
SCHEMBL337504 0.80 HCAR2 (0.89) HCAR2LMNAALDH1A1CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0731784-A1 ARYL HALIDE SUBSTITUTED METALLIC COMPLEXES, PHARMACEUTICALS CONTAINING THESE COMPLEXES, THEIR USE FOR DIAGNOSTIC PURPOSES, AND METHODS FOR PREPARING THE COMPLEXES AND PHARMACEUTICALS SCHERING AKTIENGESELLSCHAFT (DE) 1996-09-18 EP disclosed
WO-1995015306-A1 ARYL HALIDE SUBSTITUTED METALLIC COMPLEXES, PHARMACEUTICALS CONTAINING THESE COMPLEXES, THEIR USE FOR DIAGNOSTIC PURPOSES, AND METHODS FOR PREPARING THE COMPLEXES AND PHARMACEUTICALS SCHERING AKTIENGESELLSCHAFT (DE) 1995-06-08 WO disclosed