SCHEMBL9002001

SCHEMBL9002001

CCCCN(CCSc1cccc2nccn12)C(N)=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
POLB P06746 2/20 0.34
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32
GRIN2B Q13224 1/20 0.32
GRIN2C Q14957 1/20 0.32
GRIN3A Q8TCU5 1/20 0.32
ALDH1A1 P00352 2/20 0.31
HPGD P15428 1/20 0.31
CDK8 P49336 2/20 0.31
ROCK1 Q13464 2/20 0.31
FLT1 P17948 1/20 0.31
CDK9 P50750 1/20 0.31
LIMK1 P53667 1/20 0.31
CLK4 Q9HAZ1 1/20 0.31
CHEK1 O14757 1/20 0.31
MAP4K4 O95819 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9002203 0.93 SMN1; SMN2 (0.34) TP53GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL9002610 0.90 HSD17B10 (0.34) ALDH1A1HPGDCDK8ROCK1FLT1
SCHEMBL9002396 0.83 CDK8 (0.34) ALDH1A1HPGDCDK8ROCK1FLT1
SCHEMBL9002391 0.80 CDK8 (0.32) CDK8ROCK1FLT1CDK9LIMK1
SCHEMBL9002232 0.78 CDK8 (0.37) ALDH1A1HPGDCDK8ROCK1FLT1
SCHEMBL9002450 0.77 ALDH1A1 (0.33) POLBALDH1A1HPGDCDK8ROCK1
SCHEMBL9001960 0.76 CDK8 (0.34) CDK8ROCK1FLT1CDK9LIMK1
SCHEMBL9002265 0.74 ADORA2A (0.38) ALDH1A1RAB9A
SCHEMBL9189084 0.73 POLB (0.42) POLBALDH1A1HPGDMAPT
SCHEMBL9002520 0.72 ACHE (0.43) POLBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587383-A CALMODULIN INHIBITORS; ANTIISCHEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-24 US disclosed
EP-0471236-B1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-03-15 EP disclosed
US-5395839-A Calmodulin and angiogenesis inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-03-07 US disclosed
US-5244908-A Calmodulin inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-14 US disclosed
EP-0471236-A1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-02-19 EP disclosed