SCHEMBL9002409

SCHEMBL9002409

CN(C)c1cccc2c(S(=O)(=O)NCCSc3cccc4nccn34)cccc12

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 14/20 0.50
KDM4E B2RXH2 1/20 0.47
NSD2 O96028 1/20 0.47
TSHR P16473 1/20 0.47
HSD17B10 Q99714 1/20 0.47
HDAC4 P56524 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
HDAC5 Q9UQL6 1/20 0.46
HTR1A P08908 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9001942 0.85 CYP3A4 (0.45) KDM4EHSD17B10HTR1A
Hydrochloric Acid SCHEMBL9001969 0.84 SCN1A (0.46) KDM4EHSD17B10
SCHEMBL9001901 0.79 CYP3A4 (0.48) KDM4EHSD17B10HTR1A
SCHEMBL9002062 0.79 PPARG (0.37)
SCHEMBL9002030 0.78 CYP3A4 (0.50) KDM4EHSD17B10HTR1A
SCHEMBL9001992 0.78 PPARG (0.63) KDM4ETSHRHSD17B10
SCHEMBL9002172 0.78 MAPT (0.43) TSHRHSD17B10
SCHEMBL9001975 0.77 KMT2A (0.47) KDM4ETSHRHSD17B10
Hydrochloric Acid SCHEMBL9001908 0.77 MAPT (0.42) TSHRHSD17B10
SCHEMBL9002027 0.77 CNR2 (0.36) KDM4ETSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587383-A CALMODULIN INHIBITORS; ANTIISCHEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-24 US disclosed
EP-0471236-B1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-03-15 EP disclosed
US-5395839-A Calmodulin and angiogenesis inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-03-07 US disclosed
US-5244908-A Calmodulin inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-14 US disclosed
EP-0471236-A1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-02-19 EP disclosed