SCHEMBL9002995

SCHEMBL9002995

CS(=O)(=O)c1ccc(-n2nc(C(F)F)cc2-c2ccc(I)cc2)cc1

nearest known ligand 0.69

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 11/20 0.69
PTGS1 P23219 4/20 0.64
CYP2C9 P11712 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8954915 1.00 PTGS2 (0.69) PTGS2PTGS1CYP2C9
SCHEMBL8954509 0.89 PTGS2 (0.80) PTGS2PTGS1CYP2C9
SCHEMBL9003118 0.89 PTGS2 (0.73) PTGS2PTGS1
SCHEMBL8953911 0.89 PTGS2 (0.73) PTGS2PTGS1
SCHEMBL8954050 0.89 PTGS2 (0.65) PTGS2PTGS1CYP2C9
SCHEMBL8635509 0.88 PTGS2 (0.78) PTGS2PTGS1
SCHEMBL9002971 0.88 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL8953956 0.88 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL8924564 0.88 PTGS2 (0.64) PTGS2PTGS1CYP2C9
SCHEMBL3243184 0.88 PTGS2 (0.82) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0731793-A1 1,5-DIPHENYL PYRAZOLE COMPOUNDS FOR TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-09-18 EP claimed
WO-1995015315-A1 1,5-DIPHENYL PYRAZOLE COMPOUNDS FOR TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-06-08 WO claimed
EP-0731793-A1 1,5-DIPHENYL PYRAZOLE COMPOUNDS FOR TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-09-18 EP disclosed
US-5475018-A Antiinflammatory agent, antiarthritic agent; analgesics and antipyretics G. D. SEARLE & CO. (US) 1995-12-12 US disclosed
WO-1995015315-A1 1,5-DIPHENYL PYRAZOLE COMPOUNDS FOR TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-06-08 WO disclosed