SCHEMBL9003038

SCHEMBL9003038

COc1ccccc1CC(=N)N1C[C@@H]2[C@H](F)CCC(c3ccccc3)(c3ccccc3)[C@@H]2C1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 4/20 0.65
MEN1 O00255 2/20 0.65
KMT2A Q03164 2/20 0.65
CYP3A4 P08684 1/20 0.65
MAPT P10636 1/20 0.65
TSHR P16473 1/20 0.65
CYP2C19 P33261 1/20 0.65
FNTA P49354 6/20 0.56
FNTB P49356 6/20 0.56
ADRA1B P35368 3/20 0.37
HTR1A P08908 2/20 0.37
ADRA1D P25100 2/20 0.37
ADRA1A P35348 2/20 0.37
GRIN2B Q13224 1/20 0.37
CHRM3 P20309 2/20 0.34
SIGMAR1 Q99720 1/20 0.34
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34
CHRM1 P11229 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9003165 0.89 TACR1 (0.66) TACR1MEN1KMT2ACYP3A4MAPT
SCHEMBL9266283 0.88 FNTA (0.71) TACR1MEN1KMT2ACYP3A4MAPT
SCHEMBL8970958 0.88 FNTA (0.71) TACR1MEN1KMT2ACYP3A4MAPT
SCHEMBL17238244 0.82 TACR1 (0.67) TACR1MEN1KMT2ACYP3A4MAPT
SCHEMBL29407214 0.82 TACR1 (0.67) TACR1MEN1KMT2ACYP3A4MAPT
SCHEMBL4296689 0.82 TACR1 (0.67) TACR1MEN1KMT2ACYP3A4MAPT
SCHEMBL29907325 0.82 TACR1 (0.67) TACR1MEN1KMT2ACYP3A4MAPT
SCHEMBL4349316 0.78 TACR1 (1.00) TACR1MEN1KMT2ACYP3A4MAPT
SCHEMBL8460496 0.78 TACR1 (1.00) TACR1MEN1KMT2ACYP3A4MAPT
SCHEMBL7551020 0.78 TACR1 (1.00) TACR1MEN1KMT2ACYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5508433-A Derivatives of perhydroisoindole and preparation thereof RHONE-POULENC RORER S.A. (FR) 1996-04-16 US disclosed
US-5451601-A Perhydroisoindole derivatives and pharmaceutical compositions containing them RHONE-POULENC RORER S.A. (FR) 1995-09-19 US disclosed