SCHEMBL9003508

SCHEMBL9003508

C/C(N)=C(\Cc1ccccc1)C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.50
CES2 O00748 1/20 0.50
AKR1B1 P15121 1/20 0.50
HIF1A Q16665 1/20 0.46
CTBP2 P56545 1/20 0.46
ALDH1A1 P00352 3/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
TSHR P16473 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
FNTA P49354 1/20 0.42
FNTB P49356 1/20 0.42
NOS2 P35228 1/20 0.42
ALPI P09923 1/20 0.42
PKM P14618 1/20 0.42
PTGS1 P23219 1/20 0.42
XIAP P98170 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9003513 1.00 CES1 (0.50) CES1CES2AKR1B1HIF1ACTBP2
SCHEMBL5814056 0.88 CES1 (0.50) CES1CES2AKR1B1HIF1ACTBP2
SCHEMBL11109782 0.83 CES1 (0.54) CES1CES2AKR1B1CTBP2ALDH1A1
SCHEMBL3881031 0.83 CES1 (0.64) CES1CES2AKR1B1CTBP2ALDH1A1
SCHEMBL384894 0.83 CES1 (0.64) CES1CES2AKR1B1CTBP2ALDH1A1
SCHEMBL384895 0.83 CES1 (0.64) CES1CES2AKR1B1CTBP2ALDH1A1
SCHEMBL14047411 0.82 EPHX2 (0.44) CES1CES2AKR1B1HIF1AALDH1A1
SCHEMBL9003128 0.82 ALDH1A1 (0.44) CES1CES2AKR1B1HIF1AALDH1A1
SCHEMBL9003133 0.82 ALDH1A1 (0.44) CES1CES2AKR1B1HIF1AALDH1A1
SCHEMBL166471 0.82 CES1 (0.52) CES1CES2AKR1B1CTBP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0326389-B1 Process for preparing 4-hydroxypyrimidine UBE INDUSTRIES (JP) 1996-09-11 EP claimed
US-4997837-A Enzyme inhibitors WARNER-LAMBERT COMPANY (US) 1991-03-05 US disclosed
US-4906624-A 6-(((Substituted)pyridin-3-yl)alkyl)-and alkenyl)-tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis WARNER-LAMBERT COMPANY (US) 1990-03-06 US disclosed
EP-0306929-A2 6-[[(Substituted)pyridin-3-YL]alkyl]-and alkenyl]-tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis WARNER-LAMBERT COMPANY (US) 1989-03-15 EP disclosed