SCHEMBL9006337

SCHEMBL9006337

c1cnc(N2CCN(CCCOc3ccc(-c4nc5ccccc5[nH]4)cc3)CC2)nc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 11/20 1.00
DRD2 P14416 10/20 1.00
ACHE P22303 3/20 0.68
HTR1A P08908 1/20 0.58
DRD1 P21728 1/20 0.58
HTR2A P28223 1/20 0.58
HRH4 Q9H3N8 1/20 0.57
HRH3 Q9Y5N1 1/20 0.55
DRD4 P21917 1/20 0.55
LTA4H P09960 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9006318 0.90 DRD3 (1.00) DRD3DRD2ACHEHTR1ADRD1
SCHEMBL9006356 0.88 DRD3 (1.00) DRD3DRD2ACHEHTR1AHTR2A
SCHEMBL601512 0.87 DRD3 (1.00) DRD3DRD2ACHEHRH4LTA4H
SCHEMBL9260985 0.87 ACHE (0.89) DRD3DRD2ACHELTA4H
SCHEMBL5639861 0.86 ACHE (0.89) DRD3DRD2ACHEHRH3LTA4H
SCHEMBL9006372 0.85 DRD3 (0.94) DRD3DRD2ACHEHTR1AHTR2A
SCHEMBL9006339 0.85 DRD3 (1.00) DRD3DRD2ACHEHRH4DRD4
SCHEMBL9006348 0.85 DRD3 (0.85) DRD3DRD2ACHEHRH4
SCHEMBL9006359 0.85 DRD3 (0.85) DRD3DRD2ACHEHTR1ADRD1
SCHEMBL9006355 0.85 DRD3 (1.00) DRD3DRD2ACHEHTR1ADRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995030659-A1 BENZIMIDAZOLE AND IMIDAZOPYRIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS DOPAMINERGIC AGENTS, ESP. SELECTIVE FOR THE DOPAMINE D3 RECEPTOR WARNER-LAMBERT COMPANY (US) 1995-11-16 WO claimed
US-5486517-A Benzimidazoles and imidazopyridines as central nervous system agents WARNER-LAMBERT COMPANY (US) 1996-01-23 US disclosed
WO-1995030659-A1 BENZIMIDAZOLE AND IMIDAZOPYRIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS DOPAMINERGIC AGENTS, ESP. SELECTIVE FOR THE DOPAMINE D3 RECEPTOR WARNER-LAMBERT COMPANY (US) 1995-11-16 WO disclosed