SCHEMBL9260985

SCHEMBL9260985

c1ccc2[nH]c(-c3ccc(OCCCN4CCCC4)cc3)nc2c1

nearest known ligand 0.89

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ACHE P22303 6/20 0.89
DRD3 P35462 10/20 0.83
DRD2 P14416 9/20 0.78
LTA4H P09960 2/20 0.70
CHEK2 O96017 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5639861 0.99 ACHE (0.89) ACHEDRD3DRD2LTA4HCHEK2
SCHEMBL5638746 0.93 ACHE (1.00) ACHEDRD3DRD2LTA4HCHEK2
SCHEMBL601512 0.91 DRD3 (1.00) ACHEDRD3DRD2LTA4H
SCHEMBL9006356 0.88 DRD3 (1.00) ACHEDRD3DRD2
SCHEMBL9006337 0.87 DRD3 (1.00) ACHEDRD3DRD2LTA4H
SCHEMBL21017806 0.87 CHEK2 (0.72) ACHEDRD3DRD2CHEK2
SCHEMBL21018072 0.86 CHEK2 (0.74) ACHEDRD3DRD2CHEK2
SCHEMBL9006318 0.85 DRD3 (1.00) ACHEDRD3DRD2
SCHEMBL9006372 0.85 DRD3 (0.94) ACHEDRD3DRD2
SCHEMBL465443 0.85 ACHE (0.75) ACHEDRD3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995030658-A1 DIMERIC BENZIMIDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS DOPAMINERGIC AGENTS, ESP. SELECTIVE FOR THE DOPAMINE D3 RECEPTOR WARNER-LAMBERT COMPANY (US) 1995-11-16 WO disclosed
US-5414010-A Dopaminergic blocking agents and psychotic depression WARNER-LAMBERT COMPANY (US) 1995-05-09 US disclosed