SCHEMBL9006975

SCHEMBL9006975

CCOC(=O)c1ccc(C#Cc2ccc3c(c2)OC(C)(C)CC3(C)C)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 8/20 0.47
RARG P13631 6/20 0.47
RARA P10276 6/20 0.47
CYP3A4 P08684 3/20 0.47
KMT2A Q03164 2/20 0.47
CYP26A1 O43174 1/20 0.42
CRABP2 P29373 1/20 0.42
PRKCG P05129 1/20 0.39
PRKCB P05771 1/20 0.39
PRKCA P17252 1/20 0.39
PRKCE Q02156 1/20 0.39
PRKCD Q05655 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
ESR1 P03372 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
ESR2 Q92731 1/20 0.39
CA14 Q9ULX7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8624834 0.91 RARA (0.49) RARBRARGRARACYP3A4KMT2A
SCHEMBL9334969 0.89 RARA (0.62) RARBRARGRARACYP3A4KMT2A
SCHEMBL8629224 0.87 RARA (0.42) RARBRARGRARACYP3A4KMT2A
SCHEMBL9179250 0.86 RARA (0.42) RARBRARGRARACYP3A4KMT2A
SCHEMBL9180599 0.84 RARA (0.40) RARBRARGRARACYP3A4KMT2A
SCHEMBL9176298 0.84 RARA (0.40) RARBRARGRARACYP3A4KMT2A
SCHEMBL9007036 0.83 RARB (0.60) RARBRARGRARACYP3A4CYP26A1
SCHEMBL8759294 0.82 RARA (0.54) RARBRARGRARACYP3A4KMT2A
SCHEMBL9176538 0.82 RARA (0.39) RARBRARGRARACYP3A4KMT2A
SCHEMBL9329045 0.81 RARB (0.38) RARBRARGRARACYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0571546-B1 CHROMAN AND THIOCHROMANS WITH PHENYLETHYNYL SUBSTITUENTS AT THE 7-POSITION HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN INC (US) 1996-10-16 EP disclosed
US-5346915-A Chromans and thiochromans with phenylethynyl substituents at the 7-position having retinold-like biological activity ALLERGAN, INC. (US) 1994-09-13 US disclosed
EP-0571546-A1 CHROMAN AND THIOCHROMANS WITH PHENYLETHYNYL SUBSTITUENTS AT THE 7-POSITION HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY. ALLERGAN INC (US) 1993-12-01 EP disclosed
WO-1992014725-A1 CHROMAN AND THIOCHROMANS WITH PHENYLETHYNYL SUBSTITUENTS AT THE 7-POSITION HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN, INC. (US) 1992-09-03 WO disclosed