SCHEMBL9007976

SCHEMBL9007976

[CH2]c1cc([N+](=O)[O-])ccc1C

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.67
TSHR P16473 5/20 0.67
TDP1 Q9NUW8 4/20 0.67
CYP3A4 P08684 3/20 0.60
ACHE P22303 2/20 0.50
HSD17B10 Q99714 2/20 0.50
PDE2A O00408 1/20 0.50
PDE5A O76074 1/20 0.50
ALOX15 P16050 1/20 0.50
NFKB1 P19838 1/20 0.50
APEX1 P27695 1/20 0.50
PDE4A P27815 1/20 0.50
BLM P54132 1/20 0.50
PDE1B Q01064 1/20 0.50
PMP22 Q01453 1/20 0.50
PDE4B Q07343 1/20 0.50
PDE4D Q08499 1/20 0.50
PDE7A Q13946 1/20 0.50
PDE1C Q14123 1/20 0.50
PDE7B Q9NP56 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5953847 0.83 ALDH1A1 (0.67) ALDH1A1TSHRTDP1CYP3A4ACHE
SCHEMBL29511002 0.80 ALDH1A1 (1.00) ALDH1A1TSHRTDP1CYP3A4ACHE
SCHEMBL384312 0.80 ALDH1A1 (1.00) ALDH1A1TSHRTDP1CYP3A4ACHE
SCHEMBL29349558 0.77 ALDH1A1 (0.69) ALDH1A1TSHRTDP1CYP3A4ACHE
SCHEMBL10870928 0.77 TDP1 (0.61) ALDH1A1TSHRTDP1CYP3A4HSD17B10
Methylamine SCHEMBL11819150 0.77 ALDH1A1 (0.91) ALDH1A1TSHRTDP1CYP3A4ACHE
SCHEMBL2146601 0.77 GPR35 (0.59) ALDH1A1TSHRTDP1CYP3A4ACHE
SCHEMBL4400528 0.77 TSHR (0.69) ALDH1A1TSHRTDP1CYP3A4ACHE
SCHEMBL48806 0.77 ALDH1A1 (0.69) ALDH1A1TSHRTDP1CYP3A4ACHE
SCHEMBL16961844 0.76 HTT (0.48) ALDH1A1TSHRTDP1CYP3A4ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0511917-B1 Glycosylated prodrugs, process for their preparation and uses thereof HOECHST SA LAB (FR) 1996-10-23 EP claimed
WO-1992019639-A1 GLYCOSYLATED PRODRUGS, METHOD OF PREPARATION AND USE LABORATOIRES HOECHST (FR) 1992-11-12 WO claimed
EP-0511917-A1 Glycosylated prodrugs, process for their preparation and uses thereof LABORATOIRES HOECHST S.A. (FR) 1992-11-04 EP claimed
EP-2900645-A1 3-PHENYLISOXAZOLIN DERIVATIVES WITH HERBICIDAL ACTION Bayer CropScience AG (DE) 2015-08-05 EP disclosed
EP-0511917-B1 Glycosylated prodrugs, process for their preparation and uses thereof HOECHST SA LAB (FR) 1996-10-23 EP disclosed
WO-1992019639-A1 GLYCOSYLATED PRODRUGS, METHOD OF PREPARATION AND USE LABORATOIRES HOECHST (FR) 1992-11-12 WO disclosed
EP-0511917-A1 Glycosylated prodrugs, process for their preparation and uses thereof LABORATOIRES HOECHST S.A. (FR) 1992-11-04 EP disclosed
US-4029490-A BENZYLTHIOLCARBAMATE ISHIHARA SANGYO KAISHA LTD. (JA) 1977-06-14 US disclosed