SCHEMBL9010814

SCHEMBL9010814

CC(C)(NC(=O)c1cccs1)C(=O)CCl

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.56
GSK3B P49841 1/20 0.53
KDM4E B2RXH2 1/20 0.53
CASP3 P42574 1/20 0.52
CASP2 P42575 1/20 0.52
HDAC1 Q13547 2/20 0.51
GAA P10253 2/20 0.49
ALDH1A1 P00352 2/20 0.49
HDAC3 O15379 1/20 0.49
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
RAB9A P51151 6/20 0.48
NPC1 O15118 5/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
TDP1 Q9NUW8 1/20 0.47
MAPT P10636 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
HDAC11 Q96DB2 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3229709 0.83 TSHR (0.58) TSHRGSK3BKDM4ECASP3CASP2
SCHEMBL4043837 0.80 MEN1 (0.68) TSHRKDM4EHDAC1ALDH1A1MEN1
SCHEMBL30433221 0.78 TSHR (0.59) TSHRKDM4EHDAC1GAAALDH1A1
SCHEMBL9010904 0.77 TSHR (0.51) TSHRKDM4EHDAC1ALDH1A1MEN1
SCHEMBL3240216 0.76 TSHR (0.58) TSHRKDM4EHDAC1GAAALDH1A1
SCHEMBL29032333 0.75 AR (0.60) TSHRKDM4EALDH1A1MEN1KMT2A
SCHEMBL9010792 0.74 TSHR (0.55) TSHRKDM4EHDAC1GAAALDH1A1
SCHEMBL9784423 0.73 KDM4E (0.68) TSHRKDM4EHDAC1GAARAB9A
SCHEMBL29528205 0.73 CTSC (0.56) TSHRKDM4EHDAC1ALDH1A1MEN1
SCHEMBL3127881 0.73 HDAC1 (0.62) TSHRKDM4EHDAC1GAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5547984-A FUNGICIDES ROHM AND HAAS COMPANY (US) 1996-08-20 US disclosed
US-5529978-A FUNGICIDE ROHM AND HAAS COMPANY (US) 1996-06-25 US disclosed
US-5344978-A Fungicides ROHM AND HAAS COMPANY (US) 1994-09-06 US disclosed
EP-0170498-B1 N-ACETONYL-SUBSTITUTED-AMIDES, COMPOSITIONS CONTAINING THEM AND THEIR USE IN COMBATING FUNGI ROHM AND HAAS COMPANY (US) 1991-09-11 EP disclosed
US-4863940-A N-acetonyl-substituted amides and phytopathogenic fungicidal use thereof ROHM AND HAAS (US) 1989-09-05 US disclosed
EP-0170498-A2 N-acetonyl-substituted-amides, compositions containing them and their use in combating fungi ROHM AND HAAS COMPANY (US) 1986-02-05 EP disclosed