SCHEMBL9011126

SCHEMBL9011126

O=C(O)CCCc1ccccc1C1(O)CCN(C(=O)c2ccc3ccccc3c2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.47
TSHR P16473 2/20 0.47
LMNA P02545 2/20 0.47
HPGD P15428 1/20 0.46
AKR1C1 Q04828 1/20 0.46
DRD4 P21917 3/20 0.45
RAB9A P51151 1/20 0.45
S1PR5 Q9H228 1/20 0.44
CYP1A2 P05177 1/20 0.43
ALDH1A1 P00352 2/20 0.42
HTT P42858 2/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
USP2 O75604 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
ALOX15 P16050 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9011135 0.94 TSHR (0.49) NPC1TSHRLMNAHPGDAKR1C1
SCHEMBL9011001 0.87 TSHR (0.51) NPC1TSHRLMNAHPGDAKR1C1
SCHEMBL7804416 0.84 NPC1 (0.46) NPC1TSHRLMNAHPGDAKR1C1
SCHEMBL9011211 0.83 DRD4 (0.53) NPC1TSHRLMNAHPGDAKR1C1
SCHEMBL9011003 0.82 NPC1 (0.52) NPC1TSHRLMNAHPGDAKR1C1
SCHEMBL7814151 0.80 NPC1 (0.47) NPC1TSHRLMNAHPGDAKR1C1
SCHEMBL9010999 0.80 LMNA (0.59) NPC1TSHRLMNAHPGDAKR1C1
SCHEMBL9011057 0.79 NPC1 (0.52) NPC1TSHRLMNAHPGDAKR1C1
SCHEMBL7817529 0.78 PARP10 (0.51) NPC1TSHRLMNAHPGDAKR1C1
SCHEMBL9011018 0.78 NPC1 (0.54) NPC1TSHRLMNAHPGDAKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5532371-A SIDE EFFECT REDUCTION SS PHARMACEUTICAL CO., LTD. (JP) 1996-07-02 US disclosed
EP-0607536-A1 Arylamide derivatives SS PHARMACEUTICAL CO., LTD. (JP) 1994-07-27 EP disclosed