SCHEMBL9011322

SCHEMBL9011322

O=C(NCCCC(=O)C1CCCCC1)c1cnc2ccccc2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 3/20 0.57
HDAC1 Q13547 3/20 0.57
DRD2 P14416 4/20 0.51
DRD3 P35462 4/20 0.51
HTR1A P08908 2/20 0.51
HTR2A P28223 2/20 0.51
HTR2C P28335 2/20 0.51
HPGDS O60760 1/20 0.50
PREP P48147 1/20 0.50
METTL3 Q86U44 1/20 0.50
PLD2 O14939 1/20 0.47
PLD1 Q13393 1/20 0.47
KDM2B Q8NHM5 1/20 0.47
PPARD Q03181 1/20 0.46
HDAC2 Q92769 2/20 0.46
TRPV1 Q8NER1 1/20 0.46
CXCR4 P61073 1/20 0.46
HDAC4 P56524 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45
HDAC10 Q969S8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL531094 0.78 HPGDS (0.72) HPGDSTRPV1CXCR4TNKSMGAM
SCHEMBL10242977 0.78 HDAC3 (0.61) HDAC3HDAC1DRD2DRD3HTR1A
SCHEMBL5020897 0.77 HDAC3 (0.61) HDAC3HDAC1DRD2DRD3HTR1A
SCHEMBL10154201 0.77 KDM2B (0.63) HPGDSPREPMETTL3KDM2BTRPV1
Iodide SCHEMBL9011273 0.77 ACHE (0.41) HDAC3HDAC1DRD2DRD3HDAC2
SCHEMBL29222038 0.76 HDAC3 (0.61) HDAC3HDAC1DRD2DRD3HTR1A
SCHEMBL2639346 0.76 MGAM (0.56) HDAC3HDAC1DRD2DRD3HTR1A
SCHEMBL30858823 0.76 HDAC3 (0.61) HDAC3HDAC1DRD2DRD3HTR1A
SCHEMBL2639342 0.76 PPARD (0.57) HDAC3HDAC1DRD2DRD3HTR1A
SCHEMBL771034 0.75 PREP (0.59) HDAC3HDAC1DRD2DRD3HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5525727-A ANALGESIC OR NARCOTIC ANTAGONIST UNIVERSITY OF FLORIDA (US) 1996-06-11 US disclosed
US-5187158-A Sustained delivery of viricides UNIVERSITY OF FLORIDA (US) 1993-02-16 US disclosed
US-4900837-A Brain-specific drug delivery of steroid sex hormones cleaved from pyridinium carboxylates and dihydro-pyridine carboxylate precursors UNIVERSITY OF FLORIDA (US) 1990-02-13 US disclosed
US-4880921-A Brain-specific drug delivery UNIVERSITY OF FLORIDA (US) 1989-11-14 US disclosed
US-4824850-A DIHYDROPYRIDINE-PYRIDINIUM SALT REDOX CARRIER UNIVERSITY OF FLORIDA (US) 1989-04-25 US disclosed