SCHEMBL901177

SCHEMBL901177

COC(=O)CC1CCC(c2ccc(-c3ccc(-c4nc5ccc(OC)nc5[nH]4)cn3)cc2)CC1

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 20/20 0.56
KCNH2 Q12809 9/20 0.51
ADORA2A P29274 5/20 0.51
SOAT1 P35610 5/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10189192 0.93 DGAT1 (0.65) DGAT1KCNH2ADORA2ASOAT1
SCHEMBL901744 0.83 DGAT1 (0.58) DGAT1KCNH2ADORA2ASOAT1
SCHEMBL14971666 0.81 DGAT1 (0.77) DGAT1KCNH2ADORA2ASOAT1
SCHEMBL901502 0.80 DGAT1 (0.55) DGAT1KCNH2ADORA2ASOAT1
SCHEMBL10380002 0.78 DGAT1 (0.47) DGAT1KCNH2ADORA2ASOAT1
SCHEMBL15057413 0.78 DGAT1 (0.60) DGAT1KCNH2ADORA2A
SCHEMBL15057412 0.78 DGAT1 (0.60) DGAT1KCNH2ADORA2A
SCHEMBL10380275 0.78 DGAT1 (0.55) DGAT1KCNH2ADORA2ASOAT1
SCHEMBL18380764 0.78 DGAT1 (0.57) DGAT1
SCHEMBL902756 0.77 DGAT1 (0.72) DGAT1KCNH2ADORA2ASOAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed