SCHEMBL9012776

SCHEMBL9012776

O=S(=O)(c1ccc[c]c1-c1ccc(F)c(Cl)c1)C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.39
PTGS1 P23219 8/20 0.39
EPAS1 Q99814 4/20 0.36
KMO O15229 1/20 0.33
FABP4 P15090 1/20 0.32
FABP5 Q01469 1/20 0.32
GRM5 P41594 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9012933 0.90 PTGS2 (0.33) PTGS2PTGS1EPAS1KMO
SCHEMBL9012724 0.86 EPAS1 (0.34) EPAS1
SCHEMBL6401586 0.84 PTGS2 (0.50) PTGS2PTGS1
SCHEMBL9013714 0.83 PTGS2 (0.43) PTGS2PTGS1EPAS1KMO
SCHEMBL9012598 0.79 PTGS2 (0.43) PTGS2PTGS1
SCHEMBL9013024 0.75 NOTUM (0.40)
SCHEMBL9013542 0.73 PTGS2 (0.40) PTGS2PTGS1EPAS1
SCHEMBL9012951 0.73 PTGS2 (0.42) PTGS2PTGS1
SCHEMBL5790164 0.71 PTGS2 (0.41) PTGS2PTGS1
SCHEMBL27587260 0.69 PTGS2 (0.35) PTGS2PTGS1KMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0743938-A1 SUBSTITUTED SPIRO COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-11-27 EP disclosed
WO-1995021817-A1 SUBSTITUTED SPIRO COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-08-17 WO disclosed