SCHEMBL9012900

SCHEMBL9012900

NS(=O)(=O)c1ccccc1C1=C(c2ccc(O)cc2)CC2(CCCC2)C1

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.47
PTGS1 P23219 14/20 0.47
F10 P00742 2/20 0.39
SCN9A Q15858 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9012559 0.87 PTGS2 (0.47) PTGS2PTGS1
SCHEMBL9012903 0.84 PTGS2 (0.44) PTGS2PTGS1
SCHEMBL9012731 0.84 PTGS2 (0.44) PTGS2PTGS1SCN9A
SCHEMBL8386156 0.81 PTGS2 (0.69) PTGS2PTGS1
SCHEMBL8388648 0.78 PTGS2 (0.74) PTGS2PTGS1
SCHEMBL9012675 0.77 SCN9A (0.43) PTGS2PTGS1SCN9A
SCHEMBL6548544 0.75 F10 (0.52) PTGS2PTGS1F10SCN9A
SCHEMBL8384274 0.75 PTGS2 (0.72) PTGS2PTGS1
SCHEMBL8385282 0.74 PTGS2 (0.71) PTGS2PTGS1
SCHEMBL8657376 0.73 ABL1 (0.53) PTGS2PTGS1F10SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0743938-A1 SUBSTITUTED SPIRO COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-11-27 EP disclosed
WO-1995021817-A1 SUBSTITUTED SPIRO COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-08-17 WO disclosed