SCHEMBL9012903

SCHEMBL9012903

N#Cc1ccc(C2=C(c3ccccc3S(N)(=O)=O)CC3(CCCC3)C2)cc1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.44
PTGS1 P23219 9/20 0.44
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA9 Q16790 2/20 0.40
CA12 O43570 1/20 0.40
PTGES2 Q9H7Z7 2/20 0.40
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
CA13 Q8N1Q1 1/20 0.36
FABP1 P07148 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9012900 0.84 PTGS2 (0.47) PTGS2PTGS1
SCHEMBL9012559 0.84 PTGS2 (0.47) PTGS2PTGS1
SCHEMBL8384213 0.82 PTGS2 (0.64) PTGS2PTGS1CA1CA2CA9
SCHEMBL9012731 0.81 PTGS2 (0.44) PTGS2PTGS1CA2
SCHEMBL8385139 0.80 PTGS2 (0.68) PTGS2PTGS1CA1CA2CA9
SCHEMBL8385441 0.77 PTGS1 (0.67) PTGS2PTGS1CA1CA2CA9
SCHEMBL8385158 0.76 PTGS2 (0.44) PTGS2PTGS1CA1CA2CA9
SCHEMBL8659145 0.75 CA1 (0.53) PTGS2PTGS1CA1CA2CA9
SCHEMBL8384278 0.75 PTGS2 (0.68) PTGS2PTGS1
SCHEMBL9012675 0.74 SCN9A (0.43) PTGS2PTGS1CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0743938-A1 SUBSTITUTED SPIRO COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-11-27 EP disclosed
WO-1995021817-A1 SUBSTITUTED SPIRO COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-08-17 WO disclosed