SCHEMBL9013572

SCHEMBL9013572

COc1ccc(-c2cc(Cl)nc(C)n2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.53
DYRK1A Q13627 1/20 0.50
NPC1 O15118 4/20 0.49
RAB9A P51151 4/20 0.49
CXCL12 P48061 1/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
EGFR P00533 1/20 0.49
KDR P35968 1/20 0.49
AURKA O14965 1/20 0.47
AURKB Q96GD4 1/20 0.47
MAOA P21397 1/20 0.46
MAOB P27338 1/20 0.46
CASP3 P42574 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
ENPP3 O14638 1/20 0.46
ALDH1A1 P00352 3/20 0.46
MAPT P10636 3/20 0.46
HPGD P15428 3/20 0.46
ACACA Q13085 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3237986 0.87 EGFR (0.60) KDM4EDYRK1ANPC1RAB9ACXCL12
SCHEMBL3451541 0.84 KDM4E (0.67) KDM4EDYRK1ANPC1RAB9AMEN1
SCHEMBL4748830 0.82 MAPT (0.55) KDM4ECXCL12MEN1KMT2AMAOA
SCHEMBL1644753 0.81 DYRK1A (0.71) KDM4EDYRK1ANPC1RAB9AEGFR
SCHEMBL26967691 0.81 KDM4E (0.54) KDM4EDYRK1ANPC1RAB9AMEN1
SCHEMBL10686590 0.80 MEN1 (0.57) KDM4ENPC1RAB9ACXCL12MEN1
SCHEMBL25841681 0.79 NPC1 (0.59) KDM4EDYRK1ANPC1RAB9AMEN1
SCHEMBL9013563 0.79 DYRK1A (0.50) KDM4EDYRK1ANPC1RAB9ACXCL12
SCHEMBL25068057 0.79 KDM4E (0.58) KDM4ERAB9AMEN1KMT2AALDH1A1
SCHEMBL600729 0.79 RAD51 (0.44) KDM4ECXCL12MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5589477-A LEARNING ENHANCEMENT, CNS NIPPON SHINYAKU COMPANY, LIMITED (JP) 1996-12-31 US disclosed
EP-0555478-A1 PYRIMIDINE DERIVATIVE AND MEDICINE NIPPON SHINYAKU COMPANY, LIMITED (JP) 1993-08-18 EP disclosed