SCHEMBL9014174

SCHEMBL9014174

O=C(O)c1ccc(S(=O)(=O)NC(=O)c2ccc(Cl)cc2)cc1

nearest known ligand 0.87

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
FLT1 P17948 11/20 0.87
FLT4 P35916 11/20 0.87
KDR P35968 11/20 0.87
L3MBTL1 Q9Y468 1/20 0.79
PTGS1 P23219 4/20 0.69
PTGS2 P35354 4/20 0.69
EGFR P00533 2/20 0.64
BCL2L1 Q07817 1/20 0.57
MCL1 Q07820 1/20 0.57
CA1 P00915 1/20 0.57
CA2 P00918 1/20 0.57
CA9 Q16790 1/20 0.57
ALOX15 P16050 1/20 0.57
TSHR P16473 1/20 0.57
WDR5 P61964 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7287948 1.00 FLT1 (0.87) FLT1FLT4KDRL3MBTL1PTGS1
SCHEMBL10989349 0.93 FLT1 (1.00) FLT1FLT4KDRL3MBTL1PTGS1
SCHEMBL9176247 0.88 FLT1 (1.00) FLT1FLT4KDRL3MBTL1PTGS1
SCHEMBL8424044 0.86 FLT1 (0.73) FLT1FLT4KDRL3MBTL1PTGS1
SCHEMBL24224258 0.85 FLT1 (0.84) FLT1FLT4KDRL3MBTL1PTGS1
SCHEMBL9176789 0.85 FLT1 (0.84) FLT1FLT4KDRL3MBTL1PTGS1
SCHEMBL789891 0.85 FLT1 (0.84) FLT1FLT4KDRL3MBTL1PTGS1
SCHEMBL7278965 0.84 P4HTM (0.65) FLT1FLT4KDRL3MBTL1PTGS1
SCHEMBL7209929 0.83 FLT1 (0.79) FLT1FLT4KDRL3MBTL1PTGS1
SCHEMBL24224269 0.83 FLT1 (0.79) FLT1FLT4KDRL3MBTL1PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0585155-B1 Trifluoromethylketone derivatives of peptides having HLE inhibiting activity, their preparation and pharmaceutical composition ADIR (FR) 1996-12-11 EP disclosed
US-5565429-A HUMAN LEUCOCYTE ELASTASE INHIBITORS; EMPHYSEMA; ANTIARTHRITIC AGENTS; RHEUMATIC DISEASES ADIR ET COMPAGNIE (FR) 1996-10-15 US disclosed
EP-0585155-A1 Trifluoromethylketone derivatives of peptides having HLE inhibiting activity, their preparation and pharmaceutical composition ADIR ET COMPAGNIE (FR) 1994-03-02 EP disclosed