SCHEMBL8424044

SCHEMBL8424044

O=C(O)c1ccc(S(=O)(=O)NC(=O)c2ccccc2)cc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FLT1 P17948 3/20 0.73
FLT4 P35916 3/20 0.73
KDR P35968 3/20 0.73
MEN1 O00255 1/20 0.73
LMNA P02545 1/20 0.73
KMT2A Q03164 1/20 0.73
L3MBTL1 Q9Y468 1/20 0.73
BCL2L1 Q07817 4/20 0.61
MCL1 Q07820 4/20 0.61
P4HTM Q9NXG6 3/20 0.59
PTGS2 P35354 2/20 0.58
PTGS1 P23219 1/20 0.57
HTT P42858 1/20 0.55
KAT6A Q92794 1/20 0.54
ALKBH2 Q6NS38 1/20 0.54
ALKBH5 Q6P6C2 1/20 0.54
FTO Q9C0B1 1/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CA9 Q16790 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7278965 0.95 P4HTM (0.65) FLT1FLT4KDRMEN1LMNA
SCHEMBL5931288 0.89 FLT1 (0.71) FLT1FLT4KDRMEN1LMNA
SCHEMBL174010 0.89 FLT1 (0.77) FLT1FLT4KDRMEN1LMNA
Potassium SCHEMBL30358590 0.87 FLT1 (0.74) FLT1FLT4KDRMEN1LMNA
SCHEMBL29011132 0.87 FLT1 (0.74) FLT1FLT4KDRMEN1LMNA
SCHEMBL3300299 0.86 FLT1 (0.73) FLT1FLT4KDRMEN1LMNA
SCHEMBL9014174 0.86 FLT1 (0.87) FLT1FLT4KDRL3MBTL1BCL2L1
SCHEMBL9967798 0.86 FLT1 (0.69) FLT1FLT4KDRMEN1LMNA
SCHEMBL376340 0.86 MEN1 (0.73) FLT1FLT4KDRMEN1LMNA
SCHEMBL7287948 0.86 FLT1 (0.87) FLT1FLT4KDRL3MBTL1BCL2L1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5907068-A TRIFLUOROMETHYLSUBSTITUTED COMPOUND INCLUDED IN PEPTIDES ZENECA INC. (US) 1999-05-25 US disclosed
US-5726158-A INHIBITORS OF HUMAN LEUKOCYTE ELASTASE USEFUL IN TREATING TISSUE DEGENERATIVE DISEASES; TRIFLUOROMETHYL KETONE SUBSTITUTED DI-, TRI-, AND TETRA-PEPTIDE DERIVATIVES ZENECA INC. (US) 1998-03-10 US disclosed
US-5414132-A Peptide intermediates ZENECA INC. (US) 1995-05-09 US disclosed
US-5194588-A Inhibitors of human leukocyte elastase, di-, tri- and tetra-peptides ICI AMERICAS INC. (US) 1993-03-16 US disclosed
US-5055450-A Di-, tri- and tetrapeptides as inhibitors of human leukocyte elastase ICI AMERICAS INC. (US) 1991-10-08 US disclosed
US-4910190-A Containing a nitrogen containing heterocycle ring structure ICI AMERICAS INC. (US) 1990-03-20 US disclosed