SCHEMBL9014391

SCHEMBL9014391

COc1ccc(C2CCN(CCC3CCCOc4cccc(N)c43)CC2)cc1OC

nearest known ligand 0.65

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.65
DRD2 P14416 1/20 0.39
TLR9 Q9NR96 5/20 0.38
TLR7 Q9NYK1 5/20 0.38
NPSR1 Q6W5P4 1/20 0.37
TLR4 O00206 1/20 0.37
TLR3 O15455 1/20 0.37
TLR8 Q9NR97 1/20 0.37
PDE4B Q07343 2/20 0.37
QDPR P09417 1/20 0.36
HTR2C P28335 1/20 0.36
PDE4A P27815 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014647 0.92 KCNH2 (0.68) KCNH2DRD2TLR9TLR7TLR4
SCHEMBL9014660 0.89 KCNH2 (0.65) KCNH2DRD2TLR9TLR7NPSR1
SCHEMBL9015278 0.89 KCNH2 (0.65) KCNH2DRD2TLR9TLR7NPSR1
SCHEMBL9015269 0.87 KCNH2 (0.62) KCNH2DRD2TLR9TLR7TLR4
SCHEMBL9014416 0.86 KCNH2 (0.61) KCNH2DRD2PDE4BQDPR
SCHEMBL9235680 0.85 KCNH2 (0.60) KCNH2DRD2TLR9TLR7TLR4
SCHEMBL9014359 0.85 KCNH2 (0.89) KCNH2DRD2TLR9TLR7NPSR1
SCHEMBL9014644 0.84 KCNH2 (0.59) KCNH2DRD2PDE4BPDE4APDE4C
SCHEMBL9014758 0.83 KCNH2 (0.69) KCNH2DRD2TLR9TLR7TLR4
SCHEMBL9014779 0.80 KCNH2 (0.70) KCNH2DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495022-A Piperidines and piperazines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-02-27 US disclosed
EP-0634398-A1 4-Phenylpiperidinyl-1/-piperazinyl-1-ethylsubstituted benzofusedheterocycles as antiarrhythmic agents MERCK PATENT GmbH (DE) 1995-01-18 EP disclosed