SCHEMBL9014779

SCHEMBL9014779

COc1ccc2c(c1)C(CCN1CCC(c3ccc(OC)c(OC)c3)CC1)CCCO2

nearest known ligand 0.70

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.70
DRD2 P14416 3/20 0.42
ABCB1 P08183 2/20 0.42
ENPP2 Q13822 1/20 0.41
SIGMAR1 Q99720 4/20 0.40
DRD4 P21917 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014729 0.90 KCNH2 (0.69) KCNH2DRD2SIGMAR1DRD4
SCHEMBL9014758 0.90 KCNH2 (0.69) KCNH2DRD2SIGMAR1
SCHEMBL9014400 0.90 KCNH2 (0.69) KCNH2DRD2DRD4
SCHEMBL9014392 0.89 KCNH2 (0.65) KCNH2DRD2ENPP2DRD4
SCHEMBL9014359 0.89 KCNH2 (0.89) KCNH2DRD2SIGMAR1
SCHEMBL9014376 0.87 KCNH2 (0.66) KCNH2DRD2ABCB1
SCHEMBL9677908 0.84 KCNH2 (0.77) KCNH2DRD2ENPP2
Hydrochloric Acid SCHEMBL10407809 0.83 KCNH2 (0.76) KCNH2DRD2
Terikalant SCHEMBL1815992 0.82 KCNH2 (1.00) KCNH2DRD2ABCB1
Terikalant SCHEMBL30770792 0.82 KCNH2 (1.00) KCNH2DRD2ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495022-A Piperidines and piperazines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-02-27 US disclosed
EP-0634398-A1 4-Phenylpiperidinyl-1/-piperazinyl-1-ethylsubstituted benzofusedheterocycles as antiarrhythmic agents MERCK PATENT GmbH (DE) 1995-01-18 EP disclosed