SCHEMBL9014412

SCHEMBL9014412

COc1ccc(C2CCN(CCC3CCCc4cc([N+](=O)[O-])ccc43)CC2)cc1OC

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.52
DRD2 P14416 2/20 0.46
HTR2A P28223 2/20 0.46
MAPK1 P28482 1/20 0.44
SIGMAR1 Q99720 1/20 0.44
ABCB1 P08183 2/20 0.44
CCR5 P51681 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014394 0.85 KCNH2 (0.64) KCNH2DRD2HTR2AMAPK1CCR5
SCHEMBL9014667 0.85 SIGMAR1 (0.61) KCNH2SIGMAR1ABCB1
SCHEMBL9014741 0.84 KCNH2 (0.56) KCNH2SIGMAR1ABCB1
SCHEMBL9014688 0.83 KCNH2 (0.67) KCNH2DRD2SIGMAR1
SCHEMBL10407581 0.81 KCNH2 (0.71) KCNH2DRD2HTR2AMAPK1CCR5
Hydrochloric Acid SCHEMBL10407829 0.81 KCNH2 (0.70) KCNH2DRD2HTR2AMAPK1CCR5
SCHEMBL9014648 0.80 KCNH2 (0.66) KCNH2DRD2SIGMAR1
SCHEMBL9014375 0.77 KCNH2 (0.70) KCNH2DRD2SIGMAR1
SCHEMBL9235680 0.74 KCNH2 (0.60) KCNH2DRD2HTR2AMAPK1CCR5
SCHEMBL9014359 0.71 KCNH2 (0.89) KCNH2DRD2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495022-A Piperidines and piperazines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-02-27 US disclosed
EP-0634398-A1 4-Phenylpiperidinyl-1/-piperazinyl-1-ethylsubstituted benzofusedheterocycles as antiarrhythmic agents MERCK PATENT GmbH (DE) 1995-01-18 EP disclosed